CNS dejstvo

• Holecistokinin
• CCK-4
• Gastrin
• BBL-454

• Proglumid
• CI-988
• CI-1015
• L-365,260
• L-369,293
• YF-476
• YM-022
• RP-69758
• LY-225,910
• LY-288,513
• PD-135,158
• PD-145,942

• L-740,093

Povezano

Reference

1. ↑Noble F, Roques BP (July 1999). „CCK-B receptor: chemistry, molecular biology, biochemistry and pharmacology”. Prog. Neurobiol. 58 (4): 349–79. DOI:10.1016/S0301-0082(98)00090-2. PMID 10368033. 
2. ↑Pisegna JR, de Weerth A, Huppi K, Wank SA (November 1992). „Molecular cloning of the human brain and gastric cholecystokinin receptor: structure, functional expression and chromosomal localization”. Biochem. Biophys. Res. Commun. 189 (1): 296–303. DOI:10.1016/0006-291X(92)91557-7. PMID 1280419. 
3. ↑Harikumar KG, Clain J, Pinon DI, Dong M, Miller LJ (January 2005). „Distinct molecular mechanisms for agonist peptide binding to types A and B cholecystokinin receptors demonstrated using fluorescence spectroscopy”. J. Biol. Chem. 280 (2): 1044–50. DOI:10.1074/jbc.M409480200. PMID 15520004. 
4. ↑Aloj L, Caracò C, Panico M, Zannetti A, Del Vecchio S, Tesauro D, De Luca S, Arra C, Pedone C, Morelli G, Salvatore M (March 2004). „In vitro and in vivo evaluation of 111In-DTPAGlu-G-CCK8 for cholecystokinin-B receptor imaging”. J. Nucl. Med. 45 (3): 485–94. PMID 15001692. 
5. ↑Galés C, Poirot M, Taillefer J, Maigret B, Martinez J, Moroder L, Escrieut C, Pradayrol L, Fourmy D, Silvente-Poirot S (May 2003). „Identification of tyrosine 189 and asparagine 358 of the cholecystokinin 2 receptor in direct interaction with the crucial C-terminal amide of cholecystokinin by molecular modeling, site-directed mutagenesis, and structure/affinity studies”. Mol. Pharmacol. 63 (5): 973–82. DOI:10.1124/mol.63.5.973. PMID 12695525. 
6. ↑„Entrez Gene: CCKBR cholecystokinin B receptor”. 
7. ↑Altar CA, Boyar WC (April 1989). „Brain CCK-B receptors mediate the suppression of dopamine release by cholecystokinin”. Brain Res. 483 (2): 321–6. DOI:10.1016/0006-8993(89)90176-5. PMID 2706523. 
8. ↑^8,08,1Loonam TM, Noailles PA, Yu J, Zhu JP, Angulo JA (June 2003). „Substance P and cholecystokinin regulate neurochemical responses to cocaine and methamphetamine in the striatum”. Life Sci. 73 (6): 727–39. DOI:10.1016/S0024-3205(03)00393-X. PMID 12801594. 
9. ↑Lanza M, Makovec F (January 2000). „Cholecystokinin (CCK) increases GABA release in the rat anterior nucleus accumbens via CCK(B) receptors located on glutamatergic interneurons”. Naunyn Schmiedebergs Arch. Pharmacol. 361 (1): 33–8. DOI:10.1007/s002109900161. PMID 10651144. 
10. ↑Dourish CT, O'Neill MF, Coughlan J, Kitchener SJ, Hawley D, Iversen SD (January 1990). „The selective CCK-B receptor antagonist L-365,260 enhances morphine analgesia and prevents morphine tolerance in the rat”. Eur. J. Pharmacol. 176 (1): 35–44. DOI:10.1016/0014-2999(90)90129-T. PMID 2311658. 
11. ↑Higgins GA, Sills TL, Tomkins DM, Sellers EM, Vaccarino FJ (August 1994). „Evidence for the contribution of CCKB receptor mechanisms to individual differences in amphetamine-induced locomotion”. Pharmacol. Biochem. Behav. 48 (4): 1019–24. DOI:10.1016/0091-3057(94)90214-3. PMID 7972279. 
12. ↑Lu L, Huang M, Ma L, Li J (April 2001). „Different role of cholecystokinin (CCK)-A and CCK-B receptors in relapse to morphine dependence in rats”. Behav. Brain Res. 120 (1): 105–10. DOI:10.1016/S0166-4328(00)00361-2. PMID 11173090. 
13. ↑Boyce S, Rupniak NM, Tye S, Steventon MJ, Iversen SD (August 1990). „Modulatory role for CCK-B antagonists in Parkinson's disease”. Clin Neuropharmacol 13 (4): 339–47. DOI:10.1097/00002826-199008000-00009. PMID 1976438. 

Literatura

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