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UA92469C2 - Fumarate of 4-[[4-[[4-(2-cyanoethenyl)-2,6-dimethylphenyl]amino]-2-pyrimidinyl amino benzonitrile - Google Patents

Fumarate of 4-[[4-[[4-(2-cyanoethenyl)-2,6-dimethylphenyl]amino]-2-pyrimidinyl amino benzonitrile

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Publication number
UA92469C2
UA92469C2UAA200702178AUAA200702178AUA92469C2UA 92469 C2UA92469 C2UA 92469C2UA A200702178 AUAA200702178 AUA A200702178AUA A200702178 AUAA200702178 AUA A200702178AUA 92469 C2UA92469 C2UA 92469C2
Authority
UA
Ukraine
Prior art keywords
amino
cyanoethenyl
dimethylphenyl
fumarate
pyrimidinyl
Prior art date
Application number
UAA200702178A
Other languages
Russian (ru)
Inventor
Поль Теодоор Агнес Стевенс
Йозеф Пеетерс
Роже Петрус Гереберн Вандекрюйс
Альфред Элизабет Стапперс
Алекс Герман Копманс
Original Assignee
Янссен Фармацевтика Н.В.
Тиботек Фармасьютикелз Лтд.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from MYPI20043578Aexternal-prioritypatent/MY169670A/en
Application filed by Янссен Фармацевтика Н.В., Тиботек Фармасьютикелз Лтд.filedCriticalЯнссен Фармацевтика Н.В.
Publication of UA92469C2publicationCriticalpatent/UA92469C2/en

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Abstract

The present invention relates to the fumarate salt of 4-[[4-[[4-(2-cyanoethenyl)-2,6-dimethylphenyl]amino]-2-pyrimidinyl]amino]benzonitrile, pharmaceutical compositions comprising as active ingredient said salt and to processes for their preparation.
UAA200702178A2004-09-022005-09-02Fumarate of 4-[[4-[[4-(2-cyanoethenyl)-2,6-dimethylphenyl]amino]-2-pyrimidinyl amino benzonitrileUA92469C2 (en)

Applications Claiming Priority (1)

Application NumberPriority DateFiling DateTitle
MYPI20043578AMY169670A (en)2003-09-032004-09-02Combinations of a pyrimidine containing nnrti with rt inhibitors

Publications (1)

Publication NumberPublication Date
UA92469C2true UA92469C2 (en)2010-11-10

Family

ID=38137294

Family Applications (2)

Application NumberTitlePriority DateFiling Date
UAA200701971AUA92467C2 (en)2004-09-022005-09-02Hydrochloride of 4-[[4-[[4-(2-cyanoethenyl)-2,6-dimethylphenyl]amino]-2-pyrimidinyl] amino]benzonitrile
UAA200702178AUA92469C2 (en)2004-09-022005-09-02Fumarate of 4-[[4-[[4-(2-cyanoethenyl)-2,6-dimethylphenyl]amino]-2-pyrimidinyl amino benzonitrile

Family Applications Before (1)

Application NumberTitlePriority DateFiling Date
UAA200701971AUA92467C2 (en)2004-09-022005-09-02Hydrochloride of 4-[[4-[[4-(2-cyanoethenyl)-2,6-dimethylphenyl]amino]-2-pyrimidinyl] amino]benzonitrile

Country Status (6)

CountryLink
CN (2)CN101068597B (en)
AP (1)AP2296A (en)
CR (1)CR9031A (en)
SG (1)SG155885A1 (en)
UA (2)UA92467C2 (en)
ZA (1)ZA200701826B (en)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication numberPriority datePublication dateAssigneeTitle
WO2013170421A1 (en)*2012-05-142013-11-21上海迪赛诺药业有限公司Rilpivirine hydrochloride alcoholate polymorph and preparation method thereof
CN103420920B (en)*2012-05-142016-04-27上海迪赛诺药业有限公司Rilpivrine hydrochloride alcoholate polymorphic form and preparation method thereof
HRP20240118T1 (en)*2016-10-242024-04-12Janssen Sciences Ireland Unlimited CompanyDispersible compositions

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication numberPriority datePublication dateAssigneeTitle
JO3429B1 (en)*2001-08-132019-10-20Janssen Pharmaceutica NvHiv inhibiting pyrimidines derivatives
MY169670A (en)*2003-09-032019-05-08Tibotec Pharm LtdCombinations of a pyrimidine containing nnrti with rt inhibitors
PT1529032E (en)*2002-08-092013-07-11Janssen Pharmaceutica NvProcesses for the preparation of 4- 4- 4-(2 -cyanoethenyl)-2,6-dimethylphenyl )amino) -2-pyrimidinyl)amino benzonitrile

Also Published As

Publication numberPublication date
CN101068597B (en)2012-04-18
UA92467C2 (en)2010-11-10
SG155885A1 (en)2009-10-29
CR9031A (en)2009-01-16
AP2296A (en)2011-10-31
AP2007003934A0 (en)2007-04-30
CN101068597A (en)2007-11-07
CN101056673A (en)2007-10-17
ZA200701826B (en)2008-07-30

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