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SG10201606581RA - Pyrazolopyrimidinyl inhibitors of ubiquitin-activating enzyme - Google Patents

Pyrazolopyrimidinyl inhibitors of ubiquitin-activating enzyme

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Publication number
SG10201606581RA
SG10201606581RASG10201606581RASG10201606581RASG10201606581RASG 10201606581R ASG10201606581R ASG 10201606581RASG 10201606581R ASG10201606581R ASG 10201606581RASG 10201606581R ASG10201606581R ASG 10201606581RASG 10201606581R ASG10201606581R ASG 10201606581RA
Authority
SG
Singapore
Prior art keywords
ubiquitin
activating enzyme
pyrazolopyrimidinyl
inhibitors
pyrazolopyrimidinyl inhibitors
Prior art date
Application number
SG10201606581RA
Inventor
Roushan Afroze
Indu T Bharathan
Jeffrey P Ciavarri
Paul E Fleming
Jeffrey L Gaulin
Mario Girard
Steven P Langston
Francois R Soucy
Tzu-Tshin Wong
Yingchun Ye
Original Assignee
Millennium Pharm Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Millennium Pharm IncfiledCriticalMillennium Pharm Inc
Publication of SG10201606581RApublicationCriticalpatent/SG10201606581RA/en

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SG10201606581RA2012-02-172013-02-14Pyrazolopyrimidinyl inhibitors of ubiquitin-activating enzymeSG10201606581RA (en)

Applications Claiming Priority (1)

Application NumberPriority DateFiling DateTitle
US201261600070P2012-02-172012-02-17

Publications (1)

Publication NumberPublication Date
SG10201606581RAtrue SG10201606581RA (en)2016-09-29

Family

ID=48982730

Family Applications (2)

Application NumberTitlePriority DateFiling Date
SG10201606581RASG10201606581RA (en)2012-02-172013-02-14Pyrazolopyrimidinyl inhibitors of ubiquitin-activating enzyme
SG11201404757WASG11201404757WA (en)2012-02-172013-02-14Pyrazolopyrimidinyl inhibitors of ubiquitin-activating enzyme

Family Applications After (1)

Application NumberTitlePriority DateFiling Date
SG11201404757WASG11201404757WA (en)2012-02-172013-02-14Pyrazolopyrimidinyl inhibitors of ubiquitin-activating enzyme

Country Status (30)

CountryLink
US (4)US9290500B2 (en)
EP (3)EP3173413B1 (en)
JP (1)JP6122877B2 (en)
KR (1)KR20140123104A (en)
CN (1)CN104136399B (en)
AR (1)AR092797A1 (en)
BR (1)BR112014020365B1 (en)
CA (1)CA2864672C (en)
CL (1)CL2014002181A1 (en)
CO (1)CO7071135A2 (en)
CR (1)CR20140380A (en)
DO (1)DOP2014000187A (en)
EA (1)EA035020B1 (en)
EC (1)ECSP14019113A (en)
ES (1)ES2739150T3 (en)
GE (1)GEP201706687B (en)
HK (1)HK1201817A1 (en)
IL (1)IL234016A0 (en)
MA (1)MA35932B1 (en)
MX (1)MX352963B (en)
NZ (1)NZ628969A (en)
PE (1)PE20142244A1 (en)
PH (1)PH12014501832A1 (en)
SG (2)SG10201606581RA (en)
TN (1)TN2014000351A1 (en)
TW (1)TWI593688B (en)
UA (1)UA116534C2 (en)
UY (1)UY34629A (en)
WO (1)WO2013123169A1 (en)
ZA (1)ZA201406103B (en)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication numberPriority datePublication dateAssigneeTitle
US8008307B2 (en)2006-08-082011-08-30Millennium Pharmaceuticals, Inc.Heteroaryl compounds useful as inhibitors of E1 activating enzymes
KR20140123104A (en)2012-02-172014-10-21밀레니엄 파머슈티컬스 인코퍼레이티드Pyrazolopyrimidinyl inhibitors of ubiquitin-activating enzyme
WO2014022744A1 (en)2012-08-032014-02-06Millennium Pharmaceuticals, Inc.INDOLE-SUBSTITUTED PYRROLOPYRIMIDINYL INHIBITORS OF Uba6
EP3016934B1 (en)2013-07-022018-01-10Millennium Pharmaceuticals, Inc.Heteroaryl compounds useful as inhibitors of sumo activating enzyme
JP6603712B2 (en)2014-07-012019-11-06ミレニアム ファーマシューティカルズ, インコーポレイテッド Heteroaryl compounds useful as inhibitors of SUMO activating enzymes
WO2016069393A1 (en)2014-10-292016-05-06Millennium Pharmaceuticals, Inc.Administration of ubiquitin-activating enzyme inhibitor and radiation
US20180133221A1 (en)2014-10-292018-05-17Millennium Pharmaceuticals, Inc.Administration of ubiquitin-activating enzyme inhibitor and chemotherapeutic agents
AU2019370200B2 (en)2018-10-302024-12-19Kronos Bio, Inc.Compounds, compositions, and methods for modulating CDK9 activity
WO2023021498A1 (en)*2021-08-162023-02-23Moya Bio Ltd.Fused azole and furan based nucleoside analogs and uses thereof

Family Cites Families (28)

* Cited by examiner, † Cited by third party
Publication numberPriority datePublication dateAssigneeTitle
US20040023901A1 (en)2002-02-282004-02-05Cook Phillip D.Nucleoside 5'-monophosphate mimics and their prodrugs
JP2006501260A (en)2002-09-042006-01-12シェーリング コーポレイション Pyrazolopyrimidines as cyclin-dependent kinase inhibitors
US7067661B2 (en)2002-09-042006-06-27Schering CorporationPyrazolopyrimidines as cyclin dependent kinase inhibitors
US7563798B2 (en)2002-09-042009-07-21Schering CorporationSubstituted pyrazolo[1,5-a]pyrimidines as protein kinase inhibitors
US7196092B2 (en)2002-09-042007-03-27Schering CorporationN-heteroaryl pyrazolopyrimidines as cyclin dependent kinase inhibitors
WO2004087707A1 (en)2003-03-312004-10-14Vernalis (Cambridge) LimitedPyrazolopyrimidine compounds and their use in medicine
JP2005008581A (en)2003-06-202005-01-13Kissei Pharmaceut Co LtdNEW PYRAZOLO[1,5-a]PYRIMIDINE DERIVATIVE, MEDICINAL COMPOSITION CONTAINING THE SAME AND APPLICATION THEREOF
US20050130974A1 (en)2003-10-172005-06-16Rigel Pharmaceuticals, Inc.Benzothiazole compositions and their use as ubiquitin ligase inhibitors
EP1758873A1 (en)2004-06-222007-03-07Rigel Pharmaceuticals, Inc.Ubiquitin ligase inhibitors
WO2006084281A1 (en)2005-02-042006-08-10Millennium Pharmaceuticals, Inc.Inhibitors of e1 activating enzymes
WO2007044426A2 (en)2005-10-062007-04-19Schering CorporationPyrazolopyrimidines as protein kinase inhibitors
DK1989206T3 (en)2006-02-022012-10-08Millennium Pharm Inc E1 activating enzyme inhibitors
US8147618B2 (en)*2006-02-282012-04-03Lam Research AgDevice and method for liquid treating disc-like articles
MY157177A (en)2006-08-082016-05-13Millennium Pharm IncHeteroaryl compounds useful as inhibitors of e1 activating enzymes
US8008307B2 (en)2006-08-082011-08-30Millennium Pharmaceuticals, Inc.Heteroaryl compounds useful as inhibitors of E1 activating enzymes
CA2691987C (en)2007-06-122016-08-16Achaogen, Inc.Antibacterial agents
ES2757928T3 (en)2007-08-022020-04-30Millennium Pharm Inc Process for the synthesis of E1 activating enzyme inhibitors
WO2009082691A1 (en)2007-12-212009-07-02Board Of Regents, University Of Texas SystemDihydroorotate dehydrogenase inhibitors with selective anti-malarial activity
WO2010086040A1 (en)2009-01-292010-08-05Biomarin Iga, Ltd.Pyrazolo-pyrimidines for treatment of duchenne muscular dystrophy
WO2010088518A2 (en)2009-01-312010-08-05Kalypsys, Inc.Heterocyclic modulators of gpr119 for treatment of disease
NZ596470A (en)2009-05-142014-04-30Millennium Pharm IncHydrochloride salt of ((1s,2s,4r)-4-{ 4-[(1s)-2,3-dihydro-1h-inden-1-ylamino]-7h-pyrrolo [2,3-d]pyrimidin-7-yl} -2-hydroxycyclopentyl)methyl sulfamate
WO2011109059A1 (en)2010-03-012011-09-09Gtx, Inc.Compounds for treatment of cancer
US20120077814A1 (en)2010-09-102012-03-29Zhong WangSulfonamide, sulfamate, and sulfamothioate derivatives
CA2846231C (en)2011-08-242017-06-20Millennium Pharmaceuticals, Inc.Inhibitors of nedd8-activating enzyme
KR20140123104A (en)2012-02-172014-10-21밀레니엄 파머슈티컬스 인코퍼레이티드Pyrazolopyrimidinyl inhibitors of ubiquitin-activating enzyme
WO2014022744A1 (en)2012-08-032014-02-06Millennium Pharmaceuticals, Inc.INDOLE-SUBSTITUTED PYRROLOPYRIMIDINYL INHIBITORS OF Uba6
EP3016934B1 (en)2013-07-022018-01-10Millennium Pharmaceuticals, Inc.Heteroaryl compounds useful as inhibitors of sumo activating enzyme
JP6603712B2 (en)2014-07-012019-11-06ミレニアム ファーマシューティカルズ, インコーポレイテッド Heteroaryl compounds useful as inhibitors of SUMO activating enzymes

Also Published As

Publication numberPublication date
KR20140123104A (en)2014-10-21
CO7071135A2 (en)2014-09-30
TN2014000351A1 (en)2015-12-21
EP3173413A1 (en)2017-05-31
MA35932B1 (en)2014-12-01
ES2739150T3 (en)2020-01-29
CA2864672A1 (en)2013-08-22
BR112014020365B1 (en)2023-02-23
MX352963B (en)2017-12-15
CA2864672C (en)2018-01-09
US9290500B2 (en)2016-03-22
EP3536692A1 (en)2019-09-11
EP2814791A4 (en)2015-08-19
CN104136399B (en)2018-08-07
US20130217682A1 (en)2013-08-22
US9663525B2 (en)2017-05-30
US20140088096A9 (en)2014-03-27
CR20140380A (en)2014-10-28
US10202389B2 (en)2019-02-12
EP3173413B1 (en)2019-05-01
US20170217968A1 (en)2017-08-03
GEP201706687B (en)2017-06-26
UA116534C2 (en)2018-04-10
TW201345909A (en)2013-11-16
MX2014009944A (en)2014-11-10
ECSP14019113A (en)2015-09-30
DOP2014000187A (en)2014-10-15
US20160244455A1 (en)2016-08-25
JP2015508775A (en)2015-03-23
EP3536692B1 (en)2021-04-07
UY34629A (en)2013-09-02
EP2814791A1 (en)2014-12-24
EA201400831A1 (en)2014-12-30
HK1201817A1 (en)2015-09-11
PH12014501832A1 (en)2014-11-17
SG11201404757WA (en)2014-09-26
US9796725B2 (en)2017-10-24
BR112014020365A2 (en)2020-12-22
US20170369499A1 (en)2017-12-28
WO2013123169A1 (en)2013-08-22
TWI593688B (en)2017-08-01
PE20142244A1 (en)2015-01-07
AR092797A1 (en)2015-05-06
CN104136399A (en)2014-11-05
CL2014002181A1 (en)2014-12-12
IL234016A0 (en)2014-09-30
ZA201406103B (en)2017-11-29
JP6122877B2 (en)2017-04-26
NZ628969A (en)2017-03-31
EA035020B1 (en)2020-04-17

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