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MX2012007006A - Tiazoles biciclicos como moduladores alostericos de receptores mglur5. - Google Patents

Tiazoles biciclicos como moduladores alostericos de receptores mglur5.

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Publication number
MX2012007006A
MX2012007006AMX2012007006AMX2012007006AMX2012007006AMX 2012007006 AMX2012007006 AMX 2012007006AMX 2012007006 AMX2012007006 AMX 2012007006AMX 2012007006 AMX2012007006 AMX 2012007006AMX 2012007006 AMX2012007006 AMX 2012007006A
Authority
MX
Mexico
Prior art keywords
mglur5
allosteric modulators
compounds
compositions
mglur5 receptors
Prior art date
Application number
MX2012007006A
Other languages
English (en)
Inventor
Andres Avelino Trabanco-Suarez
Gregor James Macdonald
Jose Manuel Bartolome-Nebreda
Susana Conde-Ceide
Gary John Tresadern
Joaquin Pastor-Fernandez
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica NvfiledCriticalJanssen Pharmaceutica Nv
Publication of MX2012007006ApublicationCriticalpatent/MX2012007006A/es

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Abstract

La presente invención se refiere a novedosos tiazoles bicíclicos los cuales son moduladores alostéricos positivos del subtipo 5 receptor de glutamato metabotrópico ("mGluR5") y los cuales son útiles para el tratamiento o prevención de trastornos asociados con la disfunción de glutamato y enfermedades en las cuales el subtipo mGluR5 de receptores está involucrado; la invención se refiere además a composiciones farmacéuticas que comprenden dichos compuestos, a procesos para preparar dichos compuestos y composiciones, y al uso de dichos compuestos y composiciones para la prevención y tratamiento de trastornos en los cuales mGluR5 está involucrado.
MX2012007006A2009-12-182010-12-16Tiazoles biciclicos como moduladores alostericos de receptores mglur5.MX2012007006A (es)

Applications Claiming Priority (3)

Application NumberPriority DateFiling DateTitle
EP091798502009-12-18
EP101930192010-11-29
PCT/EP2010/069957WO2011073339A1 (en)2009-12-182010-12-16Bicyclic thiazoles as allosteric modulators of mglur5 receptors

Publications (1)

Publication NumberPublication Date
MX2012007006Atrue MX2012007006A (es)2012-07-03

Family

ID=43743677

Family Applications (1)

Application NumberTitlePriority DateFiling Date
MX2012007006AMX2012007006A (es)2009-12-182010-12-16Tiazoles biciclicos como moduladores alostericos de receptores mglur5.

Country Status (19)

CountryLink
US (1)US9040707B2 (es)
EP (1)EP2513117B1 (es)
JP (1)JP5763672B2 (es)
KR (1)KR20120097400A (es)
CN (1)CN102666552B (es)
AR (1)AR079509A1 (es)
AU (1)AU2010332811B2 (es)
BR (1)BR112012014436A2 (es)
CA (1)CA2782950A1 (es)
CL (1)CL2012001601A1 (es)
CO (1)CO6541615A2 (es)
EA (1)EA019980B1 (es)
ES (1)ES2431302T3 (es)
IL (1)IL220360A (es)
MX (1)MX2012007006A (es)
NZ (1)NZ600605A (es)
SG (1)SG181716A1 (es)
WO (1)WO2011073339A1 (es)
ZA (1)ZA201204433B (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication numberPriority datePublication dateAssigneeTitle
SG181715A1 (en)2009-12-182012-07-30Janssen Pharmaceutica NvBicyclic thiazoles as allosteric modulators of mglur5 receptors
ES2431302T3 (es)2009-12-182013-11-25Janssen Pharmaceutica, N.V.Tiazoles bicíclicos como moduladores alostéricos de receptores mGluR5
KR102371784B1 (ko)*2014-02-182022-03-07다이이찌 산쿄 가부시키가이샤활성화 혈액 응고 제 X 인자 (FXa) 의 저해약의 제조 방법

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US5753664A (en)*1995-03-161998-05-19Takeda Chemical Industries, Ltd.Heterocyclic compounds, their production and use
JP2002105085A (ja)*2000-09-282002-04-10Yamanouchi Pharmaceut Co Ltd新規イミダゾチアゾール誘導体
CA2503245A1 (en)*2002-10-242004-05-06Merck & Co., Inc.Alkyne derivatives as tracers for metabotropic glutamate receptor binding
TWI301760B (en)2004-02-272008-10-11Merz Pharma Gmbh & Co KgaaTetrahydroquinolinones and their use as antagonists of metabotropic glutamate receptors
JP5072602B2 (ja)2004-12-172012-11-14イーライ リリー アンド カンパニーMch受容体アンタゴニストとしてのチアゾロピリジノン誘導体
CA2593439C (en)2005-01-142014-02-25F. Hoffmann-La Roche AgThiazole-4-carboxamide derivatives as mglur5 antagonists
EP1910350A1 (en)2005-07-092008-04-16AstraZeneca AB2 -heterocyclyloxybenzoyl amino heterocyclyl compounds as modulators of glucokinase for the treatment of type 2 diabetes
WO2007023242A1 (en)*2005-08-242007-03-01Merz Pharma Gmbh & Co. KgaaTetrahydroquinolinones and their use as modulators of metabotropic glutamate receptors
KR20080059635A (ko)2005-11-072008-06-30아이알엠 엘엘씨Ppar 조절제로서의 화합물 및 조성물
RU2425834C2 (ru)*2005-11-082011-08-10Ф. Хоффманн-Ля Рош АгПРОИЗВОДНЫЕ ТИАЗОЛО[4,5-c]ПИРИДИНА В КАЧЕСТВЕ АНТАГОНИСТОВ РЕЦЕПТОРОВ mGluR5
DE102006011574A1 (de)2006-03-102007-10-31Grünenthal GmbHSubstituierte Imidazo[2,1-b]thiazol-Verbindungen und ihre Verwendung zur Herstellung von Arzneimitteln
EP2035436B1 (en)2006-06-262011-05-25UCB Pharma S.A.Fused thiazole derivatives as kinase inhibitors
WO2008012010A1 (en)2006-07-272008-01-31Ucb Pharma, S.A.Fused oxazoles & thiazoles as histamine h3- receptor ligands
GB0622202D0 (en)2006-11-072006-12-20Addex Pharmaceuticals SaNovel compounds
WO2008060597A2 (en)*2006-11-152008-05-22Vertex Pharmaceuticals IncorporatedCompounds useful as protein kinase inhibitors
JP4714669B2 (ja)2006-12-012011-06-29日本化薬株式会社ヘッダーアッシー、スクイブならびにエアバッグ用ガス発生装置およびシートベルトプリテンショナー用ガス発生装置
JP5269804B2 (ja)2006-12-142013-08-21イーライ リリー アンド カンパニー新規なmch受容体拮抗薬
EA200971143A1 (ru)2007-06-032010-06-30Вандербилт ЮниверситиБензамидные mglur5 позитивные аллостерические модуляторы и способы их получения и применения
US8642660B2 (en)*2007-12-212014-02-04The University Of RochesterMethod for altering the lifespan of eukaryotic organisms
CA2756989A1 (en)2009-04-032010-10-07Douglas BurdiCompounds for treating disorders mediated by metabotropic glutamate receptor 5, and methods of use thereof
EP2512477A4 (en)2009-12-182013-07-10Boehringer Ingelheim Int HCV POLYTHERAPY
ES2431302T3 (es)2009-12-182013-11-25Janssen Pharmaceutica, N.V.Tiazoles bicíclicos como moduladores alostéricos de receptores mGluR5

Also Published As

Publication numberPublication date
CA2782950A1 (en)2011-06-23
EP2513117B1 (en)2013-08-28
CO6541615A2 (es)2012-10-16
EA201290532A1 (ru)2012-11-30
SG181716A1 (en)2012-07-30
CN102666552B (zh)2014-11-26
IL220360A (en)2015-03-31
CN102666552A (zh)2012-09-12
ES2431302T3 (es)2013-11-25
US9040707B2 (en)2015-05-26
KR20120097400A (ko)2012-09-03
CL2012001601A1 (es)2012-10-05
JP5763672B2 (ja)2015-08-12
WO2011073339A1 (en)2011-06-23
AR079509A1 (es)2012-02-01
EP2513117A1 (en)2012-10-24
AU2010332811A1 (en)2012-06-21
JP2013514325A (ja)2013-04-25
AU2010332811B2 (en)2014-07-24
BR112012014436A2 (pt)2019-09-24
ZA201204433B (en)2014-11-26
US20120258955A1 (en)2012-10-11
NZ600605A (en)2013-08-30
EA019980B1 (ru)2014-07-30

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