FR2724654B1 - NEW GALLIC ACID DERIVATIVES, THEIR PREPARATION PROCESS, THE NEW INTERMEDIATES OBTAINED, THEIR APPLICATION AS MEDICAMENTS AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM - Google Patents

NEW GALLIC ACID DERIVATIVES, THEIR PREPARATION PROCESS, THE NEW INTERMEDIATES OBTAINED, THEIR APPLICATION AS MEDICAMENTS AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM

Info

Publication number: FR2724654B1
Authority: FR; France
Prior art keywords: new; medicaments; application; pharmaceutical compositions; preparation process
Prior art date: 1994-09-16
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Expired - Fee Related

Other versions

Inventor

Michel Fortin

Jean Luc Haesslein

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Sanofi Aventis France

Original Assignee

Roussel Uclaf SA

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1994-09-16

Filing date

1994-09-16

Publication date

1997-12-12

1994-09-16Application filed by Roussel Uclaf SAfiledCriticalRoussel Uclaf SA

1994-09-16Priority to FR9411063ApriorityCriticalpatent/FR2724654B1/en

1995-09-15Priority to PCT/FR1995/001185prioritypatent/WO1996008483A1/en

1996-03-22Publication of FR2724654A1publicationCriticalpatent/FR2724654A1/en

1997-12-12Application grantedgrantedCritical

1997-12-12Publication of FR2724654B1publicationCriticalpatent/FR2724654B1/en

2014-09-16Anticipated expirationlegal-statusCritical

StatusExpired - Fee Relatedlegal-statusCriticalCurrent

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
- C07C69/76—Esters of carboxylic acids having a carboxyl group bound to a carbon atom of a six-membered aromatic ring
- C07C69/84—Esters of carboxylic acids having a carboxyl group bound to a carbon atom of a six-membered aromatic ring of monocyclic hydroxy carboxylic acids, the hydroxy groups and the carboxyl groups of which are bound to carbon atoms of a six-membered aromatic ring
- C07C69/92—Esters of carboxylic acids having a carboxyl group bound to a carbon atom of a six-membered aromatic ring of monocyclic hydroxy carboxylic acids, the hydroxy groups and the carboxyl groups of which are bound to carbon atoms of a six-membered aromatic ring with etherified hydroxyl groups
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C233/00—Carboxylic acid amides
- C07C233/64—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings
- C07C233/81—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C309/00—Sulfonic acids; Halides, esters, or anhydrides thereof
- C07C309/63—Esters of sulfonic acids
- C07C309/64—Esters of sulfonic acids having sulfur atoms of esterified sulfo groups bound to acyclic carbon atoms
- C07C309/65—Esters of sulfonic acids having sulfur atoms of esterified sulfo groups bound to acyclic carbon atoms of a saturated carbon skeleton
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C309/00—Sulfonic acids; Halides, esters, or anhydrides thereof
- C07C309/63—Esters of sulfonic acids
- C07C309/64—Esters of sulfonic acids having sulfur atoms of esterified sulfo groups bound to acyclic carbon atoms
- C07C309/67—Esters of sulfonic acids having sulfur atoms of esterified sulfo groups bound to acyclic carbon atoms of an unsaturated carbon skeleton
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C309/00—Sulfonic acids; Halides, esters, or anhydrides thereof
- C07C309/63—Esters of sulfonic acids
- C07C309/72—Esters of sulfonic acids having sulfur atoms of esterified sulfo groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
- C07C309/73—Esters of sulfonic acids having sulfur atoms of esterified sulfo groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton to carbon atoms of non-condensed six-membered aromatic rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C309/00—Sulfonic acids; Halides, esters, or anhydrides thereof
- C07C309/63—Esters of sulfonic acids
- C07C309/72—Esters of sulfonic acids having sulfur atoms of esterified sulfo groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
- C07C309/75—Esters of sulfonic acids having sulfur atoms of esterified sulfo groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing singly-bound oxygen atoms bound to the carbon skeleton
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C309/00—Sulfonic acids; Halides, esters, or anhydrides thereof
- C07C309/63—Esters of sulfonic acids
- C07C309/72—Esters of sulfonic acids having sulfur atoms of esterified sulfo groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
- C07C309/76—Esters of sulfonic acids having sulfur atoms of esterified sulfo groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing nitrogen atoms, not being part of nitro or nitroso groups, bound to the carbon skeleton
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C309/00—Sulfonic acids; Halides, esters, or anhydrides thereof
- C07C309/63—Esters of sulfonic acids
- C07C309/72—Esters of sulfonic acids having sulfur atoms of esterified sulfo groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
- C07C309/77—Esters of sulfonic acids having sulfur atoms of esterified sulfo groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing carboxyl groups bound to the carbon skeleton
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
- C07C311/15—Sulfonamides having sulfur atoms of sulfonamide groups bound to carbon atoms of six-membered aromatic rings
- C07C311/21—Sulfonamides having sulfur atoms of sulfonamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the sulfonamide groups bound to a carbon atom of a six-membered aromatic ring
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C327/00—Thiocarboxylic acids
- C07C327/20—Esters of monothiocarboxylic acids
- C07C327/26—Esters of monothiocarboxylic acids having carbon atoms of esterified thiocarboxyl groups bound to carbon atoms of six-membered aromatic rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
- C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
- C07D317/44—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D317/46—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems condensed with one six-membered ring

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

FR9411063A1994-09-161994-09-16 NEW GALLIC ACID DERIVATIVES, THEIR PREPARATION PROCESS, THE NEW INTERMEDIATES OBTAINED, THEIR APPLICATION AS MEDICAMENTS AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEMExpired - Fee RelatedFR2724654B1 (en)

Priority Applications (2)

Application Number	Priority Date	Filing Date	Title
FR9411063AFR2724654B1 (en)	1994-09-16	1994-09-16	NEW GALLIC ACID DERIVATIVES, THEIR PREPARATION PROCESS, THE NEW INTERMEDIATES OBTAINED, THEIR APPLICATION AS MEDICAMENTS AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
PCT/FR1995/001185WO1996008483A1 (en)	1994-09-16	1995-09-15	Gallic acid derivatives, method for their preparation and their use as drugs

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
FR9411063AFR2724654B1 (en)	1994-09-16	1994-09-16	NEW GALLIC ACID DERIVATIVES, THEIR PREPARATION PROCESS, THE NEW INTERMEDIATES OBTAINED, THEIR APPLICATION AS MEDICAMENTS AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM

Publications (2)

Publication Number	Publication Date
FR2724654A1 FR2724654A1 (en)	1996-03-22
FR2724654B1true FR2724654B1 (en)	1997-12-12

Family

ID=9466996

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
FR9411063AExpired - Fee RelatedFR2724654B1 (en)	1994-09-16	1994-09-16	NEW GALLIC ACID DERIVATIVES, THEIR PREPARATION PROCESS, THE NEW INTERMEDIATES OBTAINED, THEIR APPLICATION AS MEDICAMENTS AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM

Country Status (2)

Country	Link
FR (1)	FR2724654B1 (en)
WO (1)	WO1996008483A1 (en)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US6699896B1 (en)	1998-05-12	2004-03-02	Wyeth	Oxazole-aryl-carboxylic acids useful in the treatment of insulin resistance and hyperglycemia
US6110963A (en)*	1998-05-12	2000-08-29	American Home Products Corporation	Aryl-oxo-acetic acids useful in the treatment of insulin resistance and hyperglycemia
US6063815A (en)*	1998-05-12	2000-05-16	American Home Products Corporation	Benzopenones useful in the treatment of insulin resistance and hyperglycemia
CN1308604A (en)	1998-05-12	2001-08-15	美国家用产品公司	2,3,5-substituted biphenyls useful in the treatment of insulin resistance and hyperglycemia
US6451827B2 (en)	1998-05-12	2002-09-17	Wyeth	2,3,5-substituted biphenyls useful in the treatment of insulin resistance and hyperglycemia
US6232322B1 (en)	1998-05-12	2001-05-15	American Home Products Corporation	Biphenyl oxo-acetic acids useful in the treatment of insulin resistance and hyperglycemia
US6221902B1 (en)	1998-05-12	2001-04-24	American Home Products Corporation	Biphenyl sulfonyl aryl carboxylic acids useful in the treatment of insulin resistance and hyperglycemia
US6310081B1 (en)	1999-05-10	2001-10-30	American Home Products Corporation	Biphenyl sulfonyl aryl carboxylic acids useful in the treatment of insulin resistance and hyperglycemia
NZ566263A (en)	2002-05-24	2009-09-25	Millennium Pharm Inc	CCR9 inhibitors and methods of use thereof
US7741519B2 (en)	2007-04-23	2010-06-22	Chemocentryx, Inc.	Bis-aryl sulfonamides
US7227035B2 (en)	2002-11-18	2007-06-05	Chemocentryx	Bis-aryl sulfonamides
ES2369720T5 (en)	2002-11-18	2014-11-06	Chemocentryx, Inc.	Arylsulfonamides
US7420055B2 (en)	2002-11-18	2008-09-02	Chemocentryx, Inc.	Aryl sulfonamides
US7449599B2 (en)	2004-05-13	2008-11-11	Merck + Co Inc.	Phenyl carboxamide compounds useful as beta-secretase inhibitors for the treatment of alzheimer's disease
TWI525068B (en)*	2010-09-16	2016-03-11	三菱化學股份有限公司	Novel derivative of phenolsulfonate aryl ester and thermosensitive recording material using the same
JP6184325B2 (en)*	2011-10-31	2017-08-23	日本製紙株式会社	Phenolsulfonic acid aryl ester, color developer and heat-sensitive recording material

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US2407309A (en)*	1942-02-04	1946-09-10	Squibb & Sons Inc	Chemotherapeutic agents of the sulphonamide type
DE1493482A1 (en)*	1965-06-01	1969-01-16	Boehringer Sohn Ingelheim	Process for the preparation of 3,4-dihydroxyphenylalkanolamines
NL6818531A (en)*	1968-02-09	1969-08-12
BE757005A (en)*	1969-10-02	1971-04-02	Bristol Myers Co	SUBSTITUTED PHENETHANOLAMINES AND PROCESS FOR THEIR PREPARATION
US3812194A (en)*	1970-01-06	1974-05-21	American Cyanamid Co	Novel process for preparing 6-halo-3-methylphenols
CH562199A5 (en)*	1970-10-30	1975-05-30	Hoffmann La Roche
AR206496A1 (en)*	1972-07-03	1976-07-30	Riker Laboratories Inc	PROCEDURE FOR THE PREPARATION OF 2-PHENOXY-4-NITRO-ALKYL OR HALOALKYLSULPHONANILIDES
FR2358389A1 (en)*	1976-07-15	1978-02-10	Labaz	NEW ACETOPHENONE SULPHONYL DERIVATIVES, THEIR PREPARATION PROCESS AND THEIR APPLICATIONS TO THE PREPARATION OF STABILIZERS FOR THERMOPLASTIC RESINS
US4401676A (en)*	1977-06-01	1983-08-30	Merck & Co., Inc.	Novel α-amino acids
US4507320A (en)*	1983-12-07	1985-03-26	Smithkline Beckman Corporation	Dopaminergic agonist N,N-di-n-propyl-4-hydroxy-3-methanesulfonamidophenethylamine
JPH0446175A (en)*	1990-06-14	1992-02-17	Fuji Photo Film Co Ltd	Production of 5-hydroxy-3,4-methylenedioxybenzoic acid derivative
FR2670484B1 (en)*	1990-12-18	1993-03-12	Roussel Uclaf	NEW PROCESS FOR REGIOSPECIFIC MONOFUNCTIONALIZATION OF A PHENOLIC HYDROXY ON A POLYPHENOL.
NZ247440A (en)*	1992-05-06	1995-04-27	Squibb & Sons Inc	Phenyl sulphonamide derivatives, preparation and pharmaceutical compositions thereof

1994
- 1994-09-16FRFR9411063Apatent/FR2724654B1/ennot_activeExpired - Fee Related
1995
- 1995-09-15WOPCT/FR1995/001185patent/WO1996008483A1/enactiveApplication Filing

Also Published As

Publication number	Publication date
FR2724654A1 (en)	1996-03-22
WO1996008483A1 (en)	1996-03-21

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Legal Events

Date	Code	Title
1997-04-30	CA	Change of address
1997-04-30	CD	Change of name or company name
1998-04-03	TP	Transmission of property
2001-06-29	ST	Notification of lapse

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