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FR2547587B1 - RADIOACTIVE STEROIDS, THEIR PREPARATION PROCESS, THEIR APPLICATION TO THE EVIDENCE OF GLUCOCORTICOID RECEPTORS AND TO THE DETERMINATION OF THE NUMBER OF FIXING SITES - Google Patents

RADIOACTIVE STEROIDS, THEIR PREPARATION PROCESS, THEIR APPLICATION TO THE EVIDENCE OF GLUCOCORTICOID RECEPTORS AND TO THE DETERMINATION OF THE NUMBER OF FIXING SITES

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Publication number
FR2547587B1
FR2547587B1FR8309811AFR8309811AFR2547587B1FR 2547587 B1FR2547587 B1FR 2547587B1FR 8309811 AFR8309811 AFR 8309811AFR 8309811 AFR8309811 AFR 8309811AFR 2547587 B1FR2547587 B1FR 2547587B1
Authority
FR
France
Prior art keywords
evidence
determination
application
preparation process
glucocorticoid receptors
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
FR8309811A
Other languages
French (fr)
Other versions
FR2547587A1 (en
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sanofi Aventis France
Original Assignee
Roussel Uclaf SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roussel Uclaf SAfiledCriticalRoussel Uclaf SA
Priority to FR8309811ApriorityCriticalpatent/FR2547587B1/en
Priority to NO841797Aprioritypatent/NO162193C/en
Priority to CA000456494Aprioritypatent/CA1222743A/en
Priority to AT84401202Tprioritypatent/ATE43132T1/en
Priority to FI842397Aprioritypatent/FI83784C/en
Priority to DE8484401202Tprioritypatent/DE3478225D1/en
Priority to EP84401202Aprioritypatent/EP0128839B1/en
Priority to JP59120899Aprioritypatent/JPS6034987A/en
Priority to US06/620,457prioritypatent/US4664850A/en
Publication of FR2547587A1publicationCriticalpatent/FR2547587A1/en
Application grantedgrantedCritical
Publication of FR2547587B1publicationCriticalpatent/FR2547587B1/en
Priority to US06/797,140prioritypatent/US4865767A/en
Priority to CA000529937Aprioritypatent/CA1242696A/en
Expiredlegal-statusCriticalCurrent

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Abstract

Novel radioactive steroids labelled with tritium of the formula I wherein 3H is tritium and R and R1 are individually selected from the group consisting of hydrogen, alkyl of 1 to 6 carbon atoms and acyl of an organic carboxylic acid of 1 to 10 carbon atoms useful for revealing receptors of glucocorticoids and in determining the number of fixation sites of glucocorticoids and novel intermediates.
FR8309811A1983-06-141983-06-14 RADIOACTIVE STEROIDS, THEIR PREPARATION PROCESS, THEIR APPLICATION TO THE EVIDENCE OF GLUCOCORTICOID RECEPTORS AND TO THE DETERMINATION OF THE NUMBER OF FIXING SITESExpiredFR2547587B1 (en)

Priority Applications (11)

Application NumberPriority DateFiling DateTitle
FR8309811AFR2547587B1 (en)1983-06-141983-06-14 RADIOACTIVE STEROIDS, THEIR PREPARATION PROCESS, THEIR APPLICATION TO THE EVIDENCE OF GLUCOCORTICOID RECEPTORS AND TO THE DETERMINATION OF THE NUMBER OF FIXING SITES
NO841797ANO162193C (en)1983-06-141984-05-04 RADIOACTIVE STEROID, PROCEDURE IN ITS FORECAST, Means of Detection in Vitro of GLUCOCORTICOIDER RECEIVERS FOR DETERMINING NUMBER OF GLUCOCORTICOID BINDING POINTS AND APPLICATION OF THE STEROID FOR IT
AT84401202TATE43132T1 (en)1983-06-141984-06-13 RADIOACTIVE STEROIDS, THEIR PRODUCTION, INTERMEDIATE PRODUCTS, THEIR APPLICATION TO HIGHLIGHT THE GLUCOCORTICOID RECEPTORS AND DETERMINE THE NUMBER OF BINDING SITES.
FI842397AFI83784C (en)1983-06-141984-06-13 RADIOACTIVE STEROIDER AND DERASE MELLAN PROCESSOR, FOERFARANDE FOER FRAMSTAELLNING AV DESSA OCH DERAS LAEMPLIGHET FOER PAOVISANDE AV GLUCOCORTIKOIDRECEPTORER OCH BESTAEMMANDE AV ANTALET BINDNINGSSTA.
DE8484401202TDE3478225D1 (en)1983-06-141984-06-13Labelled steroids, process for their preparation and intermediates, their use in the localization of the glucocorticoid receptors and in the dosage of the number of binding sites
EP84401202AEP0128839B1 (en)1983-06-141984-06-13Labelled steroids, process for their preparation and intermediates, their use in the localization of the glucocorticoid receptors and in the dosage of the number of binding sites
CA000456494ACA1222743A (en)1983-06-141984-06-13Radioactive steroids, preparation process and use to detect glucocorticoid receptors and for the assay of the number of fixation sites
JP59120899AJPS6034987A (en)1983-06-141984-06-14 Radioactive steroids, their production methods, and drugs for use in detecting glucocorticoid receptors and quantifying the number of fixed sites
US06/620,457US4664850A (en)1983-06-141984-06-14Novel radioactive steroids
US06/797,140US4865767A (en)1983-06-141985-12-19Novel radioactive steroids
CA000529937ACA1242696A (en)1983-06-141987-02-17Intermediates for the preparation of radioactive steroids

Applications Claiming Priority (1)

Application NumberPriority DateFiling DateTitle
FR8309811AFR2547587B1 (en)1983-06-141983-06-14 RADIOACTIVE STEROIDS, THEIR PREPARATION PROCESS, THEIR APPLICATION TO THE EVIDENCE OF GLUCOCORTICOID RECEPTORS AND TO THE DETERMINATION OF THE NUMBER OF FIXING SITES

Publications (2)

Publication NumberPublication Date
FR2547587A1 FR2547587A1 (en)1984-12-21
FR2547587B1true FR2547587B1 (en)1985-10-25

Family

ID=9289758

Family Applications (1)

Application NumberTitlePriority DateFiling Date
FR8309811AExpiredFR2547587B1 (en)1983-06-141983-06-14 RADIOACTIVE STEROIDS, THEIR PREPARATION PROCESS, THEIR APPLICATION TO THE EVIDENCE OF GLUCOCORTICOID RECEPTORS AND TO THE DETERMINATION OF THE NUMBER OF FIXING SITES

Country Status (9)

CountryLink
US (2)US4664850A (en)
EP (1)EP0128839B1 (en)
JP (1)JPS6034987A (en)
AT (1)ATE43132T1 (en)
CA (2)CA1222743A (en)
DE (1)DE3478225D1 (en)
FI (1)FI83784C (en)
FR (1)FR2547587B1 (en)
NO (1)NO162193C (en)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication numberPriority datePublication dateAssigneeTitle
FR2592047B1 (en)*1985-12-191988-03-04Roussel Uclaf ORGANOMETALLIC COMPLEXES OF STEROID PRODUCTS HAVING AFFINITY FOR THE PROGESTOGENIC AND GLUCO-CORTICOID RECEPTORS AND THEIR APPLICATION TO THE DETERMINATION OF HORMONAL RECEPTORS
ES2347027T3 (en)1998-05-222010-10-22The Board Of Trustees Of The Leland Stanford Junior University BIFUNCTIONAL MOLECULES AND THERAPIES BASED ON THE SAME.
EP3827747A1 (en)2005-04-282021-06-02Otsuka Pharmaceutical Co., Ltd.Pharma-informatics system
US9062126B2 (en)2005-09-162015-06-23Raptor Pharmaceuticals Inc.Compositions comprising receptor-associated protein (RAP) variants specific for CR-containing proteins and uses thereof
PT3395372T (en)2009-02-202022-05-05Enhanx Biopharm IncGlutathione-based drug delivery system
KR101741629B1 (en)2009-05-062017-05-31라보라토리 스킨 케어, 인크.Dermal delivery compositions comprising active agent-calcium phosphate particle complexes and methods of using the same

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication numberPriority datePublication dateAssigneeTitle
FR1465484A (en)*1965-10-271967-01-13 Ketone-type steroid compounds
FR2398077A1 (en)*1977-07-191979-02-16Roussel UclafTritiated androgenic steroid(s) - useful in the study of androgenic receptors in the body
FR2398076A1 (en)*1977-07-191979-02-16Roussel UclafTritiated nor:pregnatriene:diol, ether(s) and ester(s) - useful in the study of oestrogen receptors and tumours
FR2430952A1 (en)*1978-07-131980-02-08Roussel Uclaf NOVEL ACETYLENIC DERIVATIVES OF ANDROST 4-ENE, THEIR PREPARATION PROCESS AND THEIR APPLICATION AS A MEDICAMENT

Also Published As

Publication numberPublication date
JPS6034987A (en)1985-02-22
FI842397A0 (en)1984-06-13
ATE43132T1 (en)1989-06-15
EP0128839A3 (en)1985-09-18
CA1242696A (en)1988-10-04
US4865767A (en)1989-09-12
JPH0460479B2 (en)1992-09-28
NO162193B (en)1989-08-14
FI83784C (en)1991-08-26
FI842397L (en)1984-12-15
NO841797L (en)1984-12-17
DE3478225D1 (en)1989-06-22
EP0128839A2 (en)1984-12-19
NO162193C (en)1989-11-22
FI83784B (en)1991-05-15
US4664850A (en)1987-05-12
CA1222743A (en)1987-06-09
EP0128839B1 (en)1989-05-17
FR2547587A1 (en)1984-12-21

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DateCodeTitleDescription
CAChange of address
CDChange of name or company name
TPTransmission of property
STNotification of lapse
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