| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19843445298DE3445298A1 (en) | 1984-12-12 | 1984-12-12 | NEW PTERIDINE, METHOD FOR THE PRODUCTION AND USE THEREOF AS INTERMEDIATE PRODUCTS OR AS A MEDICINAL PRODUCT |
| DE3445298 | 1984-12-12 |
| Publication Number | Publication Date |
|---|---|
| FI854862A0true FI854862A0 (en) | 1985-12-10 |
| FI854862A7 FI854862A7 (en) | 1986-06-13 |
| FI82696B FI82696B (en) | 1990-12-31 |
| FI82696C FI82696C (en) | 1991-04-10 |
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FI854862AFI82696C (en) | 1984-12-12 | 1985-12-10 | PROCEDURE FOR THE PREPARATION OF PHARMACOLOGICAL PROPERTIES OF PTERIDINER. |
| Country | Link |
|---|---|
| EP (1) | EP0185259A3 (en) |
| JP (1) | JPS61140585A (en) |
| AU (1) | AU576924B2 (en) |
| CA (1) | CA1252783A (en) |
| DE (1) | DE3445298A1 (en) |
| DK (1) | DK161327C (en) |
| ES (1) | ES8707238A1 (en) |
| FI (1) | FI82696C (en) |
| GR (1) | GR852996B (en) |
| IL (1) | IL77294A (en) |
| NO (1) | NO161373C (en) |
| NZ (1) | NZ214522A (en) |
| PH (1) | PH24451A (en) |
| PT (1) | PT81650B (en) |
| ZA (1) | ZA859462B (en) |
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7276506B2 (en) | 1998-12-28 | 2007-10-02 | 4 Aza Bioscience Nv | Immunosuppressive effects of pteridine derivatives |
| EE200400042A (en) | 2001-06-28 | 2004-10-15 | Essential Therapeutics, Inc. | 8/17 Heterocyclic Compounds and Their Use as D-Alanyl-D-Alanine Ligase Inhibitors |
| DE10202468A1 (en)* | 2002-01-23 | 2004-09-30 | Faustus Forschungs Cie. Translational Cancer Research Gmbh | Pteridine derivatives, process for their preparation and their use |
| ES2295897T3 (en)* | 2003-08-29 | 2008-04-16 | 4 Aza Ip Nv | IMMUNODEPRESSING EFFECTS OF PTERIDINE DERIVATIVES. |
| DE602004008312T2 (en)* | 2003-10-17 | 2008-04-17 | 4 Aza Ip Nv | Heterocyclic-substituted pteridine derivatives and their use in therapy |
| GB2407089A (en)* | 2003-10-17 | 2005-04-20 | 4 Aza Bioscience Nv | Pteridine derivatives |
| JP2007526323A (en)* | 2004-03-04 | 2007-09-13 | ニューロジェン・コーポレーション | Arylalkylamino substituted quinazoline analogs |
| DE102004057594A1 (en) | 2004-11-29 | 2006-06-08 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Substitute pteridine for the treatment of inflammatory diseases |
| DE102004057618A1 (en) | 2004-11-29 | 2006-06-01 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Substituted pteridines for the treatment of inflammatory diseases |
| DE102004057595A1 (en) | 2004-11-29 | 2006-06-08 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Substituted pteridines for the treatment of inflammatory diseases |
| DE102004057645A1 (en)* | 2004-11-29 | 2006-06-01 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | New substituted pteridine compounds, useful as phosphodiesterase 4 inhibitors for treating e.g. inflammatory diseases, cancer, asthma, ulcerative colitis, depression and schizophrenia |
| JP5161102B2 (en)* | 2005-11-22 | 2013-03-13 | クドス ファーマシューティカルズ リミテッド | Pyridopyrimidine, pyrazopyrimidine and pyrimidopyrimidine derivatives as mTOR inhibitors |
| RU2445315C2 (en)* | 2005-11-22 | 2012-03-20 | Кудос Фармасьютиклз Лимитед | PYRIDO-, PYRAZO- AND PYRIMIDO-PYRIMIDINE DERIVATIVES AND USE THEREOF AS mTOR INHIBITORS |
| WO2007135026A2 (en) | 2006-05-24 | 2007-11-29 | Boehringer Ingelheim International Gmbh | Substituted pteridines as therapeutic agents |
| US10144736B2 (en) | 2006-07-20 | 2018-12-04 | Gilead Sciences, Inc. | Substituted pteridines useful for the treatment and prevention of viral infections |
| WO2008009078A2 (en) | 2006-07-20 | 2008-01-24 | Gilead Sciences, Inc. | 4,6-dl- and 2,4,6-trisubstituted quinazoline derivatives useful for treating viral infections |
| DK2057156T3 (en) | 2006-08-23 | 2017-05-08 | Kudos Pharm Ltd | 2-METHYLMORPHOLINPYRIDO, PYRAZO AND PYRIMIDO-PYRIMIDINE DERIVATIVES AS MTOR INHIBITORS |
| US8198441B2 (en) | 2008-06-20 | 2012-06-12 | Astrazeneca Ab | Process for the preparation of novel pyridopyrazines as mTOR kinase inhibitors |
| MD3097102T2 (en) | 2015-03-04 | 2018-02-28 | Gilead Sciences Inc | Toll-like receptor modulating 4,6-diamino-pyrido[3,2-D]pyrimidine compounds |
| CA3035346A1 (en) | 2016-09-02 | 2018-03-08 | Gilead Sciences, Inc. | Toll like receptor modulator compounds |
| WO2018045150A1 (en) | 2016-09-02 | 2018-03-08 | Gilead Sciences, Inc. | 4,6-diamino-pyrido[3,2-d]pyrimidine derivaties as toll like receptor modulators |
| TWI751516B (en) | 2019-04-17 | 2022-01-01 | 美商基利科學股份有限公司 | Solid forms of a toll-like receptor modulator |
| TW202212339A (en) | 2019-04-17 | 2022-04-01 | 美商基利科學股份有限公司 | Solid forms of a toll-like receptor modulator |
| TWI879779B (en) | 2019-06-28 | 2025-04-11 | 美商基利科學股份有限公司 | Processes for preparing toll-like receptor modulator compounds |
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3159628A (en)* | 1962-05-28 | 1964-12-01 | Smith Kline French Lab | Pteridine-5-oxide derivatives |
| DE3323932A1 (en)* | 1983-07-02 | 1985-01-10 | Dr. Karl Thomae Gmbh, 7950 Biberach | NEW 2-PIPERAZINO-PTERIDINE, METHOD FOR THE PRODUCTION THEREOF AND MEDICINAL PRODUCTS CONTAINING THIS COMPOUND |
| Publication number | Publication date |
|---|---|
| ES8707238A1 (en) | 1987-07-16 |
| FI854862A7 (en) | 1986-06-13 |
| DK161327B (en) | 1991-06-24 |
| NO854965L (en) | 1986-06-13 |
| PH24451A (en) | 1990-06-25 |
| FI82696B (en) | 1990-12-31 |
| DK572685A (en) | 1986-06-13 |
| NZ214522A (en) | 1988-07-28 |
| IL77294A (en) | 1989-02-28 |
| DK161327C (en) | 1991-12-09 |
| DE3445298A1 (en) | 1986-06-12 |
| NO161373B (en) | 1989-05-02 |
| ZA859462B (en) | 1987-07-29 |
| EP0185259A3 (en) | 1989-03-01 |
| DK572685D0 (en) | 1985-12-11 |
| AU5123285A (en) | 1986-06-19 |
| PT81650A (en) | 1986-01-01 |
| AU576924B2 (en) | 1988-09-08 |
| ES549806A0 (en) | 1987-07-16 |
| CA1252783A (en) | 1989-04-18 |
| JPS61140585A (en) | 1986-06-27 |
| FI82696C (en) | 1991-04-10 |
| EP0185259A2 (en) | 1986-06-25 |
| GR852996B (en) | 1986-04-16 |
| PT81650B (en) | 1988-04-21 |
| NO161373C (en) | 1989-08-09 |
| Publication | Publication Date | Title |
|---|---|---|
| FI855102A7 (en) | TETRAHYDRO-BENZTHIAZOLER, DERAS FRAMSTAELLNING OCH DERAS ANVAENDNING SAOSOM MELLANPRODUKTER ELLER SAOSOM LAEKEMEDEL. | |
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| Date | Code | Title | Description |
|---|---|---|---|
| MM | Patent lapsed | Owner name:DR. KARL THOMAE GESELLSCHAFT MIT |