Movatterモバイル変換


[0]ホーム

URL:


ECSP982601A - INDOL COMPOUNDS AS ANTI-INFLAMMATORY / ANALGESIC AGENTS - Google Patents

INDOL COMPOUNDS AS ANTI-INFLAMMATORY / ANALGESIC AGENTS

Info

Publication number
ECSP982601A
ECSP982601AECSP982601AECSP982601AEC SP982601 AECSP982601 AEC SP982601AEC SP982601 AECSP982601 AEC SP982601AEC SP982601 AECSP982601 AEC SP982601A
Authority
EC
Ecuador
Prior art keywords
hydrogen
4alkyl
inflammatory
analgesic agents
4alkoxy
Prior art date
Application number
Other languages
Spanish (es)
Inventor
Kazunari Nakao
Chikara Uchida
Kiyoshi Kawamura
Rodney William Stevens
Shinya Fujiwara
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filedfiledCritical
Priority to ECSP982601priorityCriticalpatent/ECSP982601A/en
Publication of ECSP982601ApublicationCriticalpatent/ECSP982601A/en

Links

Landscapes

Abstract

Translated fromSpanish

Esta invención proporciona un compuesto de la siguiente fórmula: (gráfico), y las sales farmacéuticamente aceptables del mismo, en la que L es oxígeno o azufre; y es un enlace directo o alquilideno C1-4; Q es alquilo C1-6; cicloalquilo C3-7, fenilo naftilo, heteroarilo o similares; R1 es hidrógeno, alquilo C1-6 o similares; R2 es hidrógeno, alquilo C1-4, C(O)R5 donde R5 es alquilo C1-22 o alquenilo C2-22, alquilo C1-8 halosustituido, alquenilo C2-8 halosustituido -y- cicloalquilo C3-7 -y-cicloalquenilo C3-7 -y- cicloalquenilo C3-7, fenilo naftilo, heteroarilo o similares X es halo alquilo C1-4, hidroxi alcoxi C1-4 p similares; X es halo, alquilo C1-4, hidroxi, alcoxi C1-4 o similares; y n es o 1,2 ó 3 con la condición de que un grupo de fórmula -y-Q no es metilo o etilo cuando X es hidrógeno; L es oxigeno; R1 es hidrógeno; y R2 es acetilo. Esta invención también proporciona una composición farmacéutica útil para el tratamiento de una afección médica en la que estan implicadas lasprostaglandinas como patógenos.This invention provides a compound of the following formula: (graph), and the pharmaceutically acceptable salts thereof, wherein L is oxygen or sulfur; y is a direct bond or C1-4alkylidene; Q is C1-6alkyl; C3-7cycloalkyl, phenyl naphthyl, heteroaryl or the like; R1 is hydrogen, C1-6 alkyl or the like; R2 is hydrogen, C1-4alkyl, C (O) R5 where R5 is C1-22alkyl or C2-22alkenyl, halosubstituted C1-8alkyl, C2-8alkenylhalosubstituted -y- C3-7cycloalkyl-C3 -7 -y- C3-7cycloalkenyl, phenyl naphthyl, heteroaryl, or the like X is halo C1-4alkyl, hydroxy C1-4alkoxy, or the like; X is halo, C1-4alkyl, hydroxy, C1-4alkoxy, or the like; and n is either 1,2 or 3 with the proviso that a group of the formula -y-Q is not methyl or ethyl when X is hydrogen; L is oxygen; R1 is hydrogen; and R2 is acetyl. This invention also provides a pharmaceutical composition useful for the treatment of a medical condition in which lasprostaglandins are implicated as pathogens.

ECSP9826011998-07-221998-07-22 INDOL COMPOUNDS AS ANTI-INFLAMMATORY / ANALGESIC AGENTSECSP982601A (en)

Priority Applications (1)

Application NumberPriority DateFiling DateTitle
ECSP982601ECSP982601A (en)1998-07-221998-07-22 INDOL COMPOUNDS AS ANTI-INFLAMMATORY / ANALGESIC AGENTS

Applications Claiming Priority (1)

Application NumberPriority DateFiling DateTitle
ECSP982601ECSP982601A (en)1998-07-221998-07-22 INDOL COMPOUNDS AS ANTI-INFLAMMATORY / ANALGESIC AGENTS

Publications (1)

Publication NumberPublication Date
ECSP982601Atrue ECSP982601A (en)1999-02-11

Family

ID=42043521

Family Applications (1)

Application NumberTitlePriority DateFiling Date
ECSP982601ECSP982601A (en)1998-07-221998-07-22 INDOL COMPOUNDS AS ANTI-INFLAMMATORY / ANALGESIC AGENTS

Country Status (1)

CountryLink
EC (1)ECSP982601A (en)

Similar Documents

PublicationPublication DateTitle
CO4810382A1 (en) INDOL COMPOUNDS ANTI-INFLAMMATORY / ANALGESICAL AGENTS
AR035617A1 (en) COMPOUNDS DERIVED FROM PHENETHANOLAMINE, COMBINATIONS AND PHARMACEUTICAL FORMULATIONS OF THE SAME, PROCESS FOR THEIR PREPARATION, ITS USE IN THE PREPARATION OF MEDICINES FOR THE TREATMENT OR PROPHYLAXIS OF A CLINICAL CONDITION FOR WHICH A BETAIEPAR BARDIAR AGENT IS ADDED
ECSP034563A (en) IMIDAZOL COMPOUNDS CONDENSED WITH ARILO OR HETEROARILO AS ANTI-INFLAMMATORY AND ANALGESIC AGENTS
DE60142891D1 (en) AZETIDINE DERIVATIVES PHARMACEUTICAL COMPOSITIONS, THE AZETIDINE DERIVATIVES AND THEIR PREPARATION
PA8466201A1 (en) INDOL 2,3-SUBSTITUTED COMPOUNDS AS ANTI-INFLAMMATORY AND ANALGESIC AGENTS
CY1107853T1 (en) APPLICABLE AMINOXIC USES FOR THE TREATMENT OF BIPHICAL DISORDERS
DK1065204T3 (en) Bicyclic carbonyl indole compounds as anti-inflammatory / analgesic agents and as COX-2 inhibitors
AR035812A1 (en) PHARMACEUTICALLY EFFECTIVE ACRILAMIDE COMPOUNDS AS INHIBITORS OF THE ENOIL-ACP REDUCTASA-FABI-; COMPOSITIONS FORMULATED WITH SUCH COMPOUNDS, METHOD FOR INHIBITING SUCH REDUCTION, RESPECTIVELY, TO TREAT BACTERIAL INFECTIONS USING SUCH COMPOUNDS AND USE OF THE COMPOUNDS MENCI
AR055613A1 (en) CRYSTAL FORMS DELTA AND EPSILON OF IMATINIB MESILATE
AR047076A1 (en) PIRROLOTRIAZINE COMPOUNDS AS THYROSINE KINASE INHIBITORS, PHARMACEUTICAL COMPOSITIONS
PL369108A1 (en)17beta-hydroxysteroid dehydrogenase type 3 inhibitors for the treatment of androgen dependent diseases
UY30025A1 (en) SUBSTITUTED DERIVATIVES OF 2-AMINO-5,6-DIHIDRO PIRIMIDIN-4 (3H) -ONAS AND ITS PHARMACEUTICALLY ACCEPTABLE SALTS, PHARMACEUTICAL COMPOSITIONS CONTAINING AND APPLICATIONS.
PE20040728A1 (en) CASPASE INHIBITORS
ES2421948T3 (en) Compounds and compositions for delivering active agents
ATE305777T1 (en) AGENT FOR PREVENTING CHRONIC REJECTION REACTION AS A RESULT OF ORGAN TRANSPLANTATION
HN2002000110A (en) USE OF (Z) - 2 - CIANO - 3 - HYDROXY - BUTIL - 2 - ENOIC ACID (4 '- TRIFLUOROMETIL PHENYL) - AMIDA FOR THE TREATMENT OF MULTIPLE SCLEROSIS.
UY38971A (en) HETEROCYCLIC COMPOUNDS AS DELTA-5 DESATURASE INHIBITORS AND METHODS OF USE
TR200302106T4 (en) N-benzenesulfonyl L-Proline compounds as antagonists of bradykinin
AR037250A1 (en) COMPOSITE OF 1H-QUINOLIN-2-ONA REPLACED, PROCESS FOR PREPARATION, MEDICATION THAT INCLUDES IT AND ITS USE IN THE MANUFACTURE OF A MEDICINAL PRODUCT
ECSP982601A (en) INDOL COMPOUNDS AS ANTI-INFLAMMATORY / ANALGESIC AGENTS
AR033779A1 (en) USEFUL COMPOUNDS IN REFLUX DISEASE
CR9417A (en) 7-FLUORO-1,3-DIHIDRO-INDOL-2-ONA OXAZOLIDINONES AS ANTIBACTERIAL AGENTS
AR050101A1 (en) OXAZOLIDINONES CONTAINING OXINDOLS AS ANTIBACTERIAL AGENTS.
DE602005017629D1 (en) PHARMACEUTICAL COMPOSITIONS FOR THE TREATMENT OF LEISHMANIASIS
UY26741A1 (en) HYGROMYCIN A DERIVATIVES

[8]ページ先頭

©2009-2025 Movatter.jp