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DK340387A - acyl derivatives - Google Patents

acyl derivatives

Info

Publication number
DK340387A
DK340387ADK340387ADK340387ADK340387ADK 340387 ADK340387 ADK 340387ADK 340387 ADK340387 ADK 340387ADK 340387 ADK340387 ADK 340387ADK 340387 ADK340387 ADK 340387A
Authority
DK
Denmark
Prior art keywords
represents hydrogen
halogen
group
lower alkyl
salts
Prior art date
Application number
DK340387A
Other languages
Danish (da)
Other versions
DK340387D0 (en
Inventor
Harry Allen Albrecht
Ka-Kong Chan
Dennis Dalton Keith
Rudolf Ludwig Then
Manfred Weigele
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La RochefiledCriticalHoffmann La Roche
Publication of DK340387D0publicationCriticalpatent/DK340387D0/en
Publication of DK340387ApublicationCriticalpatent/DK340387A/en

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Abstract

Cephalosporin derivatives of the formula <IMAGE> in which m represents 0, 1 or 2, R<1> represents hydrogen or an acyl group, R<2> represents hydrogen, lower alkoxy, amino, lower alkylthio or lower alkanoylamino, R<3><1> represents hydrogen, lower alkyl, lower alkenyl, C3-C7-cycloalkyl, halogen-lower alkyl or halophenyl; Z represents R<3><0>-C or nitrogen, R<3><0> represents hydrogen or halogen, or R<3><0> and R<3><1> together represent a C3-C5-alkylene group, a C2-C4-alkylene- monooxy group or a C1-C2-alkylenedioxy group, R<3><2> represents hydrogen, halogen, lower alkyl or an optionally substituted 5- or 6-membered heterocyclic ring having one, two or three oxygen, nitrogen and/or sulphur atoms and R<3><3> represents hydrogen or halogen or R<3><2> and R<3><3> together represent a C1-C4-alkylenedioxy group, and easily hydrolysable esters and salts of these compounds and hydrates of the compounds of the formula I or of their esters and salts are described. The products have antimicrobial activity.
DK340387A1986-07-031987-07-02 acyl derivativesDK340387A (en)

Applications Claiming Priority (1)

Application NumberPriority DateFiling DateTitle
US88155586A1986-07-031986-07-03

Publications (2)

Publication NumberPublication Date
DK340387D0 DK340387D0 (en)1987-07-02
DK340387Atrue DK340387A (en)1988-01-04

Family

ID=25378717

Family Applications (1)

Application NumberTitlePriority DateFiling Date
DK340387ADK340387A (en)1986-07-031987-07-02 acyl derivatives

Country Status (22)

CountryLink
EP (1)EP0251330B1 (en)
JP (1)JPH0730083B2 (en)
KR (1)KR880001675A (en)
CN (1)CN1021226C (en)
AT (2)ATE97901T1 (en)
AU (1)AU603364B2 (en)
CS (2)CS270227B2 (en)
DE (1)DE3788306D1 (en)
DK (1)DK340387A (en)
ES (1)ES2060583T3 (en)
FI (1)FI88392C (en)
HU (1)HU200185B (en)
IE (1)IE61434B1 (en)
IL (1)IL83046A (en)
MC (1)MC1833A1 (en)
MX (1)MX7189A (en)
NO (1)NO168890C (en)
NZ (1)NZ220914A (en)
PH (1)PH23940A (en)
PT (1)PT85246B (en)
ZA (1)ZA874696B (en)
ZW (1)ZW12787A1 (en)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication numberPriority datePublication dateAssigneeTitle
NZ227470A (en)*1987-12-281991-06-25Hoffmann La RocheAcyl derivatives of substituted cephem compounds; pharmaceutical compositions and methods for preparation and treatment
YU63689A (en)*1988-03-311991-06-30Hoffmann La RocheAcyl derivatives
CA2001203C (en)*1988-10-242001-02-13Thomas P. Demuth, Jr.Novel antimicrobial dithiocarbamoyl quinolones
ES2129388T3 (en)*1988-10-241999-06-16Procter & Gamble Pharma FLUOROQUINOLONIL-CEFEMS ANTIMICROBIALS.
EP0997466A1 (en)*1988-10-242000-05-03PROCTER &amp; GAMBLE PHARMACEUTICALS, INC.Novel antimicrobial lactam-quinolones
US5328908A (en)*1988-10-241994-07-12Procter & Gamble Pharmaceuticals, Inc.Antimicrobial quinolone thioureas
EP0366193A3 (en)*1988-10-241992-01-08Norwich Eaton Pharmaceuticals, Inc.Novel antimicrobial quinolonyl lactams
ATE194353T1 (en)*1988-10-242000-07-15Norwich Eaton Pharma ANTIMICROBIAL QUINOLONYLLACTAMESTERS
AU633867B2 (en)*1989-02-021993-02-11Eli Lilly And CompanyDelivery of cytotoxic agents
GB8907617D0 (en)*1989-04-051989-05-17Celltech LtdDrug delivery system
ATE193890T1 (en)*1990-04-182000-06-15Procter & Gamble Pharma ANTIMICROBIAL QUINOLONYL LACTAMES
US5066800A (en)*1990-04-271991-11-19Hoffmann-La Roche Inc.Qunoline intermediates useful therein for synthesizing antibacterial compounds
US5244892A (en)*1990-10-161993-09-14Kyorin Pharmaceutical Co., Ltd.Cephem compounds, and antibacterial agents
GB9216759D0 (en)*1992-08-071992-09-23Finpael SpaProcess for the production of 7-amino thiazolyl cephalosporins
DE4234330A1 (en)*1992-10-121994-04-14Bayer Ag Quinolonecarboxylic acids
ATE179422T1 (en)*1994-02-251999-05-15Aranda Lab Sa De Cv CHINOLONYLCARBOXAMIDOCEPHALOSPORINE DERIVATIVES AND MEDICINAL PRODUCTS CONTAINING SAME
MX9505113A (en)*1995-12-071997-06-28Aranda Lab Sa De CvCephalosporine-fluoroquinolonates derivatives and pharmaceutical compositions containing them.
EP3698793A1 (en)2014-01-292020-08-26Vyome Therapeutics LimitedBesifloxacin for the treatment of resistant acne

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication numberPriority datePublication dateAssigneeTitle
US3971778A (en)1972-05-121976-07-27Glaxo Laboratories LimitedCephalosporins having (α-etherified oximino)acylamido groups at the 7-position
CA1006521A (en)*1972-12-181977-03-08Minoru SugitaPiperazine derivatives and process for preparing them
US4173199A (en)1974-12-021979-11-06Codama Holding S.A.Apparatus for reinforcing a fabric by applying a fluid reinforcing material thereto
DE2760123C2 (en)1976-01-231986-04-30Roussel-Uclaf, Paris 7-Aminothiazolyl-syn-oxyiminoacetamidocephalosporanic acids, their preparation and pharmaceutical compositions containing them
DE2716677C2 (en)1977-04-151985-10-10Hoechst Ag, 6230 Frankfurt Cephem derivatives and processes for their preparation
JPS5854157B2 (en)1977-06-101983-12-02山之内製薬株式会社 New derivatives of cephalosporin compounds and their production method
JPS5630964A (en)*1979-08-221981-03-28Kyorin Pharmaceut Co LtdNovel substituted quinolinecarboxylic acid and its preparation
US4266049A (en)1980-02-201981-05-05Eli Lilly And CompanyProcess for 3-iodomethyl cephalosporins
FR2501209B1 (en)*1981-03-031986-07-04Sanofi Sa NOVEL CEPHALOSPORIN DERIVATIVES AND ANTIBIOTIC DRUGS CONTAINING THE SAME
SE440354B (en)*1981-02-191985-07-29Kyorin Seiyaku Kk quinolinecarboxylic
FR2570702B1 (en)*1984-09-271987-01-09Sanofi Sa CEPHALOSPORIN DERIVATIVES, PROCESSES FOR OBTAINING THEM AND THEIR APPLICATION AS ANTIBIOTICS
NZ214864A (en)*1985-01-211988-04-29Sankei Yakuhin Kk#b#-lactam compounds
NZ227470A (en)*1987-12-281991-06-25Hoffmann La RocheAcyl derivatives of substituted cephem compounds; pharmaceutical compositions and methods for preparation and treatment

Also Published As

Publication numberPublication date
ATE97901T1 (en)1993-12-15
PT85246B (en)1990-03-30
NO872770D0 (en)1987-07-02
PT85246A (en)1987-08-01
MC1833A1 (en)1988-06-03
PH23940A (en)1990-01-23
FI872951A7 (en)1988-01-04
HUT44258A (en)1988-02-29
CS395091A3 (en)1992-12-16
DK340387D0 (en)1987-07-02
NO872770L (en)1988-01-04
NO168890C (en)1992-04-15
IE871765L (en)1988-01-03
HU200185B (en)1990-04-28
CN87105204A (en)1988-06-29
CN1021226C (en)1993-06-16
FI88392B (en)1993-01-29
NZ220914A (en)1990-09-26
FI872951A0 (en)1987-07-03
EP0251330B1 (en)1993-12-01
ES2060583T3 (en)1994-12-01
EP0251330A2 (en)1988-01-07
IL83046A0 (en)1987-12-31
IE61434B1 (en)1994-11-02
FI88392C (en)1993-05-10
ZW12787A1 (en)1988-02-03
MX7189A (en)1993-08-01
DE3788306D1 (en)1994-01-13
AT391137B (en)1990-08-27
ATA264587A (en)1990-02-15
AU603364B2 (en)1990-11-15
AU7500987A (en)1988-01-07
ZA874696B (en)1988-01-04
IL83046A (en)1992-07-15
EP0251330A3 (en)1989-06-28
JPS6322586A (en)1988-01-30
KR880001675A (en)1988-04-26
JPH0730083B2 (en)1995-04-05
CS270227B2 (en)1990-06-13
NO168890B (en)1992-01-06
CS496787A2 (en)1989-10-13

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