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AU2003280680A1 - Xanthine compound - Google Patents

Xanthine compound

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Publication number
AU2003280680A1
AU2003280680A1AU2003280680AAU2003280680AAU2003280680A1AU 2003280680 A1AU2003280680 A1AU 2003280680A1AU 2003280680 AAU2003280680 AAU 2003280680AAU 2003280680 AAU2003280680 AAU 2003280680AAU 2003280680 A1AU2003280680 A1AU 2003280680A1
Authority
AU
Australia
Prior art keywords
xanthine compound
xanthine
compound
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU2003280680A
Inventor
Hitoshi Hochigai
Hiroyuki Nakahira
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sumitomo Pharma Co Ltd
Original Assignee
Sumitomo Pharmaceuticals Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sumitomo Pharmaceuticals Co LtdfiledCriticalSumitomo Pharmaceuticals Co Ltd
Publication of AU2003280680A1publicationCriticalpatent/AU2003280680A1/en
Abandonedlegal-statusCriticalCurrent

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AU2003280680A2002-11-012003-10-31Xanthine compoundAbandonedAU2003280680A1 (en)

Applications Claiming Priority (11)

Application NumberPriority DateFiling DateTitle
JP2002-3202162002-11-01
JP20023202162002-11-01
JP2002-3629532002-12-13
JP20023629532002-12-13
JP2002-3648852002-12-17
JP20023648852002-12-17
JP2002-3672602002-12-18
JP20023672602002-12-18
JP20023811612002-12-27
JP2002-3811612002-12-27
PCT/JP2003/013990WO2004048379A1 (en)2002-11-012003-10-31Xanthine compound

Publications (1)

Publication NumberPublication Date
AU2003280680A1true AU2003280680A1 (en)2004-06-18

Family

ID=32398335

Family Applications (1)

Application NumberTitlePriority DateFiling Date
AU2003280680AAbandonedAU2003280680A1 (en)2002-11-012003-10-31Xanthine compound

Country Status (2)

CountryLink
AU (1)AU2003280680A1 (en)
WO (1)WO2004048379A1 (en)

Cited By (23)

* Cited by examiner, † Cited by third party
Publication numberPriority datePublication dateAssigneeTitle
US8637530B2 (en)2005-07-302014-01-28Boehringer Ingelheim International Gmbh8-(3-amino-piperidin-1-yl)-xanthines, their preparation, and their use as pharmaceuticals
US8664232B2 (en)2002-08-212014-03-04Boehringer Ingelheim Pharma Gmbh & Co. Kg8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions
US8673927B2 (en)2006-05-042014-03-18Boehringer Ingelheim International GmbhUses of DPP-IV inhibitors
US8697868B2 (en)2004-02-182014-04-15Boehringer Ingelheim International Gmbh8-[3-amino-piperidin-1-yl]-xanthines, their preparation and their use as pharmaceutical compositions
US8846695B2 (en)2009-01-072014-09-30Boehringer Ingelheim International GmbhTreatment for diabetes in patients with inadequate glycemic control despite metformin therapy comprising a DPP-IV inhibitor
US8853156B2 (en)2008-08-062014-10-07Boehringer Ingelheim International GmbhTreatment for diabetes in patients inappropriate for metformin therapy
US8865729B2 (en)2008-12-232014-10-21Boehringer Ingelheim International GmbhSalt forms of a xanthine compound
US8883800B2 (en)2011-07-152014-11-11Boehringer Ingelheim International GmbhSubstituted quinazolines, the preparation thereof and the use thereof in pharmaceutical compositions
US8883805B2 (en)2004-11-052014-11-11Boehringer Ingelheim International GmbhProcess for the preparation of chiral 8-(3-aminopiperidin-1-yl)-xanthines
US9034883B2 (en)2010-11-152015-05-19Boehringer Ingelheim International GmbhVasoprotective and cardioprotective antidiabetic therapy
US9149478B2 (en)2010-06-242015-10-06Boehringer Ingelheim International GmbhDiabetes therapy
US9155705B2 (en)2008-04-032015-10-13Boehringer Ingelheim International GmbhDPP-IV inhibitor combined with a further antidiabetic agent, tablets comprising such formulations, their use and process for their preparation
US9186392B2 (en)2010-05-052015-11-17Boehringer Ingelheim International GmbhCombination therapy
US9266888B2 (en)2006-05-042016-02-23Boehringer Ingelheim International GmbhPolymorphs
US9457029B2 (en)2009-11-272016-10-04Boehringer Ingelheim International GmbhTreatment of genotyped diabetic patients with DPP-IV inhibitors such as linagliptin
US9486526B2 (en)2008-08-062016-11-08Boehringer Ingelheim International GmbhTreatment for diabetes in patients inappropriate for metformin therapy
US9526730B2 (en)2012-05-142016-12-27Boehringer Ingelheim International GmbhUse of a DPP-4 inhibitor in podocytes related disorders and/or nephrotic syndrome
US9526728B2 (en)2014-02-282016-12-27Boehringer Ingelheim International GmbhMedical use of a DPP-4 inhibitor
US9555001B2 (en)2012-03-072017-01-31Boehringer Ingelheim International GmbhPharmaceutical composition and uses thereof
US9713618B2 (en)2012-05-242017-07-25Boehringer Ingelheim International GmbhMethod for modifying food intake and regulating food preference with a DPP-4 inhibitor
US10155000B2 (en)2016-06-102018-12-18Boehringer Ingelheim International GmbhMedical use of pharmaceutical combination or composition
US11033552B2 (en)2006-05-042021-06-15Boehringer Ingelheim International GmbhDPP IV inhibitor formulations
US11911388B2 (en)2008-10-162024-02-27Boehringer Ingelheim International GmbhTreatment for diabetes in patients with insufficient glycemic control despite therapy with an oral or non-oral antidiabetic drug

Families Citing this family (35)

* Cited by examiner, † Cited by third party
Publication numberPriority datePublication dateAssigneeTitle
US7074923B2 (en)*2002-05-312006-07-11Schering CorporationProcess for preparing xanthine phosphodiesterase V inhibitors and precursors thereof
US7569574B2 (en)2002-08-222009-08-04Boehringer Ingelheim Pharma Gmbh & Co. KgPurine derivatives, the preparation thereof and their use as pharmaceutical compositions
US7495005B2 (en)2002-08-222009-02-24Boehringer Ingelheim Pharma Gmbh & Co. KgXanthine derivatives, their preparation and their use in pharmaceutical compositions
US7482337B2 (en)2002-11-082009-01-27Boehringer Ingelheim Pharma Gmbh & Co. KgXanthine derivatives, the preparation thereof and their use as pharmaceutical compositions
DE10254304A1 (en)2002-11-212004-06-03Boehringer Ingelheim Pharma Gmbh & Co. Kg New xanthine derivatives, their production and their use as medicines
US7566707B2 (en)2003-06-182009-07-28Boehringer Ingelheim International GmbhImidazopyridazinone and imidazopyridone derivatives, the preparation thereof and their use as pharmaceutical compositions
DE10355304A1 (en)2003-11-272005-06-23Boehringer Ingelheim Pharma Gmbh & Co. Kg Novel 8- (piperazin-1-yl) and 8 - ([1,4] diazepan-1-yl) xanthines, their preparation and their use as pharmaceuticals
EP2119717B1 (en)2004-02-182018-01-17Boehringer Ingelheim International GmbH8-[3-amino-piperidin-1-yl]-xanthins, their production and utilisation as DPP IV inhibitors
DE102004009039A1 (en)2004-02-232005-09-08Boehringer Ingelheim Pharma Gmbh & Co. Kg 8- [3-Amino-piperidin-1-yl] xanthines, their preparation and use as pharmaceuticals
US7393847B2 (en)2004-03-132008-07-01Boehringer Ingleheim International GmbhImidazopyridazinediones, their preparation and their use as pharmaceutical compositions
US7439370B2 (en)2004-05-102008-10-21Boehringer Ingelheim International GmbhImidazole derivatives, their preparation and their use as intermediates for the preparation of pharmaceutical compositions and pesticides
DE102004030502A1 (en)2004-06-242006-01-12Boehringer Ingelheim Pharma Gmbh & Co. Kg Novel imidazoles and triazoles, their preparation and use as medicines
DE102004037554A1 (en)2004-08-032006-03-16Sanofi-Aventis Deutschland Gmbh Substituted 8-aminoalkylthio-xanthines, process for their preparation and their use as medicaments
DE102004039507A1 (en)2004-08-142006-03-02Sanofi-Aventis Deutschland Gmbh Substituted 8-aminoalkoxi-xanthines, process for their preparation and their use as medicaments
DE102004043944A1 (en)2004-09-112006-03-30Boehringer Ingelheim Pharma Gmbh & Co. Kg Novel 8- (3-amino-piperidin-1-yl) -7- (but-2-ynyl) -xanthines, their preparation and their use as pharmaceuticals
DE102004044221A1 (en)2004-09-142006-03-16Boehringer Ingelheim Pharma Gmbh & Co. Kg New 3-methyl-7-butynyl xanthines, their preparation and their use as pharmaceuticals
AU2005292134B2 (en)*2004-10-012010-12-23Merck Sharp & Dohme Corp.Aminopiperidines as dipeptidyl peptidase-IV inhibitors for the treatment or prevention of diabetes
DOP2006000008A (en)2005-01-102006-08-31Arena Pharm Inc COMBINED THERAPY FOR THE TREATMENT OF DIABETES AND RELATED AFFECTIONS AND FOR THE TREATMENT OF AFFECTIONS THAT IMPROVE THROUGH AN INCREASE IN THE BLOOD CONCENTRATION OF GLP-1
PE20071221A1 (en)2006-04-112007-12-14Arena Pharm Inc GPR119 RECEPTOR AGONISTS IN METHODS TO INCREASE BONE MASS AND TO TREAT OSTEOPOROSIS AND OTHER CONDITIONS CHARACTERIZED BY LOW BONE MASS, AND COMBINED THERAPY RELATED TO THESE AGONISTS
WO2008017670A1 (en)2006-08-082008-02-14Boehringer Ingelheim International GmbhPyrrolo [3, 2 -d] pyrimidines as dpp-iv inhibitors for the treatment of diabetes mellitus
ES2733348T3 (en)2007-08-172019-11-28Boehringer Ingelheim Int Purine derivatives for use in the treatment of diseases related to FAP
EP2108960A1 (en)2008-04-072009-10-14Arena Pharmaceuticals, Inc.Methods of using A G protein-coupled receptor to identify peptide YY (PYY) secretagogues and compounds useful in the treatment of conditons modulated by PYY
AU2009290911A1 (en)2008-09-102010-03-18Boehringer Ingelheim International GmbhCombination therapy for the treatment of diabetes and related conditions
AR077642A1 (en)2009-07-092011-09-14Arena Pharm Inc METABOLISM MODULATORS AND THE TREATMENT OF DISORDERS RELATED TO THE SAME
JP2013523819A (en)2010-04-062013-06-17アリーナ ファーマシューティカルズ, インコーポレイテッド GPR119 receptor modulators and treatment of disorders related thereto
AU2011305525B2 (en)2010-09-222016-08-18Arena Pharmaceuticals, Inc.Modulators of the GPR119 receptor and the treatment of disorders related thereto
WO2012135570A1 (en)2011-04-012012-10-04Arena Pharmaceuticals, Inc.Modulators of the gpr119 receptor and the treatment of disorders related thereto
US20140066369A1 (en)2011-04-192014-03-06Arena Pharmaceuticals, Inc.Modulators Of The GPR119 Receptor And The Treatment Of Disorders Related Thereto
WO2012145603A1 (en)2011-04-222012-10-26Arena Pharmaceuticals, Inc.Modulators of the gpr119 receptor and the treatment of disorders related thereto
WO2012145604A1 (en)2011-04-222012-10-26Arena Pharmaceuticals, Inc.Modulators of the gpr119 receptor and the treatment of disorders related thereto
WO2012170702A1 (en)2011-06-082012-12-13Arena Pharmaceuticals, Inc.Modulators of the gpr119 receptor and the treatment of disorders related thereto
WO2013055910A1 (en)2011-10-122013-04-18Arena Pharmaceuticals, Inc.Modulators of the gpr119 receptor and the treatment of disorders related thereto
WO2014074668A1 (en)2012-11-082014-05-15Arena Pharmaceuticals, Inc.Modulators of gpr119 and the treatment of disorders related thereto
KR20180006881A (en)2015-03-092018-01-19인테크린 테라퓨틱스, 아이엔씨. Methods for the treatment of nonalcoholic fatty liver disease and / or fat dystrophy
KR20200036808A (en)2017-04-032020-04-07코히러스 바이오사이언시스, 인크. PPARγ agonist for the treatment of advanced nuclear paralysis

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication numberPriority datePublication dateAssigneeTitle
MXPA02012272A (en)*2000-07-042003-04-25Novo Nordisk AsHeterocyclic compounds, which are inhibitors of the enzyme dpp-iv.
SK286975B6 (en)*2001-02-242009-08-06Boehringer Ingelheim Pharma Gmbh & Co. KgXanthine derivatives, method the production thereof, pharmaceutical formulation containing thereof and their use
JP2005502624A (en)*2001-07-032005-01-27ノボ ノルディスク アクティーゼルスカブ Purine derivatives inhibiting DPP-IV for the treatment of diabetes

Cited By (52)

* Cited by examiner, † Cited by third party
Publication numberPriority datePublication dateAssigneeTitle
US9108964B2 (en)2002-08-212015-08-18Boehringer Ingelheim International Gmbh8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions
US8664232B2 (en)2002-08-212014-03-04Boehringer Ingelheim Pharma Gmbh & Co. Kg8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions
US10023574B2 (en)2002-08-212018-07-17Boehringer Ingelheim International Gmbh8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions
US9556175B2 (en)2002-08-212017-01-31Boehringer Ingelheim International Gmbh8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and thier use as pharmaceutical compositions
US10202383B2 (en)2002-08-212019-02-12Boehringer Ingelheim International Gmbh8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions
US9321791B2 (en)2002-08-212016-04-26Boehringer Ingelheim International Gmbh8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions
US8697868B2 (en)2004-02-182014-04-15Boehringer Ingelheim International Gmbh8-[3-amino-piperidin-1-yl]-xanthines, their preparation and their use as pharmaceutical compositions
US9751855B2 (en)2004-11-052017-09-05Boehringer Ingelheim International GmbhProcess for the preparation of chiral 8-(3-aminopiperidin-1-yl)-xanthines
US9499546B2 (en)2004-11-052016-11-22Boehringer Ingelheim International GmbhProcess for the preparation of chiral 8-(3-aminopiperidin-1-yl)-xanthines
US8883805B2 (en)2004-11-052014-11-11Boehringer Ingelheim International GmbhProcess for the preparation of chiral 8-(3-aminopiperidin-1-yl)-xanthines
US8637530B2 (en)2005-07-302014-01-28Boehringer Ingelheim International Gmbh8-(3-amino-piperidin-1-yl)-xanthines, their preparation, and their use as pharmaceuticals
US11919903B2 (en)2006-05-042024-03-05Boehringer Ingelheim International GmbhPolymorphs
US11291668B2 (en)2006-05-042022-04-05Boehringer Ingelheim International GmbhUses of DPP IV inhibitors
US8673927B2 (en)2006-05-042014-03-18Boehringer Ingelheim International GmbhUses of DPP-IV inhibitors
US9173859B2 (en)2006-05-042015-11-03Boehringer Ingelheim International GmbhUses of DPP IV inhibitors
US9815837B2 (en)2006-05-042017-11-14Boehringer Ingelheim International GmbhPolymorphs
US10301313B2 (en)2006-05-042019-05-28Boehringer Ingelheim International GmbhPolymorphs
US12171767B2 (en)2006-05-042024-12-24Boehringer Ingelheim International GmbhUses of DPP IV inhibitors
US9266888B2 (en)2006-05-042016-02-23Boehringer Ingelheim International GmbhPolymorphs
US11084819B2 (en)2006-05-042021-08-10Boehringer Ingelheim International GmbhPolymorphs
US10080754B2 (en)2006-05-042018-09-25Boehringer Ingelheim International GmbhUses of DPP IV inhibitors
US12178819B2 (en)2006-05-042024-12-31Boehringer Ingelheim International GmbhDPP IV inhibitor formulations
US11033552B2 (en)2006-05-042021-06-15Boehringer Ingelheim International GmbhDPP IV inhibitor formulations
US9493462B2 (en)2006-05-042016-11-15Boehringer Ingelheim International GmbhPolymorphs
US10973827B2 (en)2008-04-032021-04-13Boehringer Ingelheim International GmbhDPP-IV inhibitor combined with a further antidiabetic agent, tablets comprising such formulations, their use and process for their preparation
US9415016B2 (en)2008-04-032016-08-16Boehringer Ingelheim International GmbhDPP-IV inhibitor combined with a further antidiabetic agent, tablets comprising such formulations, their use and process for their preparation
US10022379B2 (en)2008-04-032018-07-17Boehringer Ingelheim International GmbhDPP-IV inhibitor combined with a further antidiabetic agent, tablets comprising such formulations, their use and process for their preparation
US9155705B2 (en)2008-04-032015-10-13Boehringer Ingelheim International GmbhDPP-IV inhibitor combined with a further antidiabetic agent, tablets comprising such formulations, their use and process for their preparation
US10034877B2 (en)2008-08-062018-07-31Boehringer Ingelheim International GmbhTreatment for diabetes in patients inappropriate for metformin therapy
US8853156B2 (en)2008-08-062014-10-07Boehringer Ingelheim International GmbhTreatment for diabetes in patients inappropriate for metformin therapy
US9486526B2 (en)2008-08-062016-11-08Boehringer Ingelheim International GmbhTreatment for diabetes in patients inappropriate for metformin therapy
US11911388B2 (en)2008-10-162024-02-27Boehringer Ingelheim International GmbhTreatment for diabetes in patients with insufficient glycemic control despite therapy with an oral or non-oral antidiabetic drug
US9212183B2 (en)2008-12-232015-12-15Boehringer Ingelheim International GmbhSalt forms of 1-[(4-methyl-quinazolin-2-yl)methyl]-3-methyl-7-(2-butyn-1-yl)-8-(3-(R)-amino-piperidin-1-yl)-xanthine
US8865729B2 (en)2008-12-232014-10-21Boehringer Ingelheim International GmbhSalt forms of a xanthine compound
US8846695B2 (en)2009-01-072014-09-30Boehringer Ingelheim International GmbhTreatment for diabetes in patients with inadequate glycemic control despite metformin therapy comprising a DPP-IV inhibitor
US9457029B2 (en)2009-11-272016-10-04Boehringer Ingelheim International GmbhTreatment of genotyped diabetic patients with DPP-IV inhibitors such as linagliptin
US10092571B2 (en)2009-11-272018-10-09Boehringer Ingelheim International GmbhTreatment of genotyped diabetic patients with DPP-IV inhibitors such as linagliptin
US10004747B2 (en)2010-05-052018-06-26Boehringer Ingelheim International GmbhCombination therapy
US9603851B2 (en)2010-05-052017-03-28Boehringer Ingelheim International GmbhCombination therapy
US9186392B2 (en)2010-05-052015-11-17Boehringer Ingelheim International GmbhCombination therapy
US9149478B2 (en)2010-06-242015-10-06Boehringer Ingelheim International GmbhDiabetes therapy
US11911387B2 (en)2010-11-152024-02-27Boehringer Ingelheim International GmbhVasoprotective and cardioprotective antidiabetic therapy
US9034883B2 (en)2010-11-152015-05-19Boehringer Ingelheim International GmbhVasoprotective and cardioprotective antidiabetic therapy
US8962636B2 (en)2011-07-152015-02-24Boehringer Ingelheim International GmbhSubstituted quinazolines, the preparation thereof and the use thereof in pharmaceutical compositions
US9199998B2 (en)2011-07-152015-12-01Boehringer Ingelheim Internatioal GmbhSubstituted quinazolines, the preparation thereof and the use thereof in pharmaceutical compositions
US8883800B2 (en)2011-07-152014-11-11Boehringer Ingelheim International GmbhSubstituted quinazolines, the preparation thereof and the use thereof in pharmaceutical compositions
US9555001B2 (en)2012-03-072017-01-31Boehringer Ingelheim International GmbhPharmaceutical composition and uses thereof
US9526730B2 (en)2012-05-142016-12-27Boehringer Ingelheim International GmbhUse of a DPP-4 inhibitor in podocytes related disorders and/or nephrotic syndrome
US10195203B2 (en)2012-05-142019-02-05Boehringr Ingelheim International GmbHUse of a DPP-4 inhibitor in podocytes related disorders and/or nephrotic syndrome
US9713618B2 (en)2012-05-242017-07-25Boehringer Ingelheim International GmbhMethod for modifying food intake and regulating food preference with a DPP-4 inhibitor
US9526728B2 (en)2014-02-282016-12-27Boehringer Ingelheim International GmbhMedical use of a DPP-4 inhibitor
US10155000B2 (en)2016-06-102018-12-18Boehringer Ingelheim International GmbhMedical use of pharmaceutical combination or composition

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