This is alist of knowncombinedsex-hormonalformulations. Brand names and developmental code names are in parentheses.
Androgens and estrogens
[edit]- Chlorotrianisene/methyltestosterone (Tace mit Androgen)[1]
- Conjugated estrogens/methyltestosterone (Premarin with Methyltestosterone)
- Dienestrol/methyltestosterone (Estan, Lucidon)
- Dienestrol diacetate/methyltestosterone (Farmatest)
- Diethylstilbestrol/methyltestosterone (Tylosterone)
- Esterified estrogens/methyltestosterone (Covaryx, Eemt, Essian, Estratest, Menogen, Syntest)
- Ethinylestradiol/methyltestosterone (Climatone, Dumone, Duotrone, Estandron, Femandren, Femovirin, Gynetone, Lynandron, Mepilin, Mixogen, Primodian)[1][2]
- Methylestradiol/methyltestosterone (Klimanosid)[2]
- Methylestradiol/methyltestosterone/reserpine (Klimanosid R)[1]
- Estradiol benzoate/testosterone propionate (Bothermon)
- Estradiol benzoate/estradiol dienanthate/testosterone enanthate benzilic acid hydrazone (Climacteron, Lactimex, Lactostat)
- Estradiol benzoate/estradiol phenylpropionate/testosterone propionate/testosterone phenylpropionate/testosterone isocaproate (Estandron Prolongatum, Lynandron Prolongatum, Mixogen [Injection])
- Estradiol benzoate/testosterone isobutyrate (Femandren M, Folivirin)
- Estradiol butyrylacetate/testosterone ketolaurate/reserpine (Klimanosid R-Depot)
- Estradiol cypionate/testosterone cypionate (Depo-Testadiol, Femovirin)
- Estradiol cypionate/testosterone enanthate (Supligol)
- Estradiol valerate/prasterone enanthate (Binodian Depot, Cidodian Depot, Gynodian Depot, Klimax, Supligol NF)
- Estradiol valerate/testosterone enanthate (Deladumone, Despamen, Ditate, Ditate-DS, Gravignost, Primodian Depot, Valertest)
Estrogens and progestogens
[edit]Inbirth control pills:
- Drospirenone/estetrol (Nextstellis, Drovelis, Lydisilka)
- Estradiol/nomegestrol acetate (Naemis, Zoely)
- Estradiol valerate/cyproterone acetate (Femilar)
- Estradiol valerate/dienogest (Natazia, Qlaira)
- Ethinylestradiol/chlormadinone acetate (Belara)[3]
- Ethinylestradiol/cyproterone acetate (Diane, Diane-35)
- Ethinylestradiol/desogestrel (Alenvona, Apri,[4] Azurette,[5] Bekyree,[6] Bimizza,[7] Caziant,[8] Cesia,[9] Cimizt,[10] Cyclessa,[11] Cyred,[12] Denise, Desogen,[13] Desirett, Emoquette,[14] Enskyce,[15] Gedarel, Gracial, Isibloom,[16] Juleber,[17] Kalliga, Kariva,[18] Kimidess,[19] Laurina, Linessa, Marvelon,[20][21][22] Mercilon,[23][24] Mircette,[25] Mirvala, Novynette, Ortho-Cept,[26] Pimtrea,[27] Reclipsen,[28] Regulon, Simliya,[29] Solia, Velivet,[30] Viorele,[31] Volnea[32])
- Ethinylestradiol/dienogest (Valette)
- Ethinylestradiol/dimethisterone (Oracon)
- Ethinylestradiol/drospirenone (Yasmin, Yasminelle, Yaz)
- Ethinylestradiol/drospirenone/levomefolic acid (Beyaz, Safyral)
- Ethinylestradiol/etynodiol diacetate (Demulen)
- Ethinylestradiol/gestodene (Femodene, Femodette, Gynera, Harmonet, Meliane, Minesse, Minulet)
- Ethinylestradiol/levonorgestrel (Amethyst, Aviane, Balcoltra, Falmina, Levlen, Lillow, Orsythia, Vienva)
- Ethinylestradiol/levonorgestrel/bisglycinate
- Ethinylestradiol/levonorgestrel/ferrous fumarate
- Ethinylestradiol/lynestrenol (Lyndiol)
- Ethinylestradiol/medroxyprogesterone acetate (Gianda, Provest)
- Ethinylestradiol/megestrol acetate (Nuvacon, Volidan)
- Ethinylestradiol/norethisterone (Brevicon, Norinyl 1+35, Ortho-Novum 7/7/7, Taytulla, Tri-Norinyl, Zenchent)
- Ethinylestradiol/norethisterone/ferrous fumarate (Blisovi 24 FE, Estrostep Fe, Femcon FE, Kaitlib FE, Lo Minastrin Fe, Loestrin 24 Fe, Microgestin 24 FE)
- Ethinylestradiol/norethisterone acetate (FemHRT)
- Ethinylestradiol/norethisterone acetate/ferrous fumarate
- Ethinylestradiol/norgestimate (Ortho Tri-Cyclen, Sprintec)
- Ethinylestradiol/norgestrel (Ovral)
- Ethinylestradiol/norgestrienone (Miniplanor, Planor)
- Ethinylestradiol/quingestanol acetate (Riglovis)
- Ethinylestradiol sulfonate/norethisterone acetate (Deposiston)
- Mestranol/anagestone acetate (Neo-Novum)
- Mestranol/chlormadinone acetate (C-Quens, Lutedion)
- Mestranol/etynodiol diacetate (Ovulen)
- Mestranol/hydroxyprogesterone acetate (Hormolidin)
- Mestranol/lynestrenol (Lyndiol)
- Mestranol/norethisterone (Norethin, Noriday, Norinyl, Norquen, Ortho-Novum)
- Mestranol/noretynodrel (Enavid, Enovid)
- Quinestrol/etynodiol diacetate (Soluna)
- Quinestrol/levonorgestrel (Yuèkětíng, Àiyuè)
- Quinestrol/norgestrel (Compound Norgestrel)
- Quinestrol/quingestanol acetate (Unovis)
Formenopausal hormone therapy and/orgynecological disorders:
- Conjugated estrogens/medrogestone (Presomen)
- Conjugated estrogens/medroxyprogesterone acetate (Prempro, Premphase)
- Conjugated estrogens/norgestrel (Prempak-C)
- Estradiol/drospirenone (Angeliq)
- Estradiol/dydrogesterone (Femoston)
- Estradiol/gestodene (Avaden, Avadene)
- Estradiol/levonorgestrel
- Estradiol/medroxyprogesterone acetate (Indivina, Tridestra)
- Estradiol/norethisterone acetate (Activella, Activelle, Cliane, Estalis, Eviana, Evorel, Kliogest, Novofem)
- Estradiol/norgestimate (Prefest)
- Estradiol/progesterone (Bijuva)
- Estradiol/trimegestone (Lovelle, Totelle)
- Estradiol valerate/cyproterone acetate (Climen, Climen 28)
- Estradiol valerate/estriol/levonorgestrel (CycloÖstrogynal)
- Estradiol valerate/levonorgestrel (Cyclo-Progynova N)
- Estradiol valerate/medroxyprogesterone acetate (Dilena, Divina, Divitren, Farludiol, Indivina, Sisare)
- Estradiol valerate/norethisterone (Climagest, Climesse)
- Estradiol valerate/norethisterone acetate (Cliovelle, Norestin, Trisequens)
- Estradiol valerate/norgestrel (Cyclacur, Cyclocur, Cyclo-Progynova, Postoval, Progyluton)
- Ethinylestradiol/ethisterone (Amenorone, Di-Pro, Duosterone, Menstrogen, Oracecron, Orasecron)[2][1]
- Mestranol/noretynodrel (Enovid)
Never or not yet marketed
[edit]Inbirth control pills:
Incontraceptive patches:
Formenopausal hormone therapy:
Incontraceptive vaginal rings:
Incombined injectable contraceptives:
- Estradiol/megestrol acetate (Mego-E, Chinese Injectable No. 2)
- Estradiol benzoate/estradiol valerate/hydroxyprogesterone caproate (Sin-Ol)
- Estradiol benzoate butyrate/algestone acetophenide (Redimen, Soluna, Unijab)
- Estradiol cypionate/hydroxyprogesterone caproate (Sinbios)
- Estradiol cypionate/medroxyprogesterone acetate (Cyclo-Provera, Cyclofem, Lunelle)
- Estradiol enanthate/algestone acetophenide (Anafertin, Deladroxate, Perlutan, Topasel, Yectames)
- Estradiol valerate/hydroxyprogesterone caproate (Chinese Injectable No. 1)
- Estradiol valerate/norethisterone enanthate (Mesigyna, Mesygest)
Formenopausal hormone therapy,gynecological disorders,habitual abortion, and other indications:
Incombined injectable contraceptives:
For other indications:
Androgens and progestogens
[edit]Estrogens, progestogens, and androgens
[edit]- ^abcdefghijHans Hermann Julius Hager; Walther Kern; Paul Heinz List; Hermann Josef Roth (29 July 2013).Hagers Handbuch der Pharmazeutischen Praxis: Für Apotheker, Arzneimittelhersteller, Ärzte und Medizinalbeamte: Wirkstoffgruppen II Chemikalien und Drogen (A-AL). Springer-Verlag. pp. 143,185–187.ISBN 978-3-662-25655-8.Archived from the original on 6 September 2022. Retrieved3 June 2019.
- ^abcdeGeorg Arends; Heinrich Zörnig; Hermann Hager; Georg Frerichs, Walther Kern (14 December 2013).Hagers Handbuch der pharmazeutischen Praxis: Für Apotheker, Arzneimittelhersteller, Drogisten, Ärzte u. Medizinalbeamte. Springer-Verlag. pp. 1163–1164.ISBN 978-3-662-36329-4.Archived from the original on 6 September 2022. Retrieved3 June 2019.
- ^"Archived copy"(PDF).Archived(PDF) from the original on 2022-09-06. Retrieved2022-09-06.
{{cite web}}: CS1 maint: archived copy as title (link) - ^"Apri 28 Day- desogestrel and ethinyl estradiol kit".DailyMed.Archived from the original on 10 July 2021. Retrieved10 July 2021.
- ^"Azurette- desogestrel/ethinyl estradiol and ethinyl estradiol kit".DailyMed.Archived from the original on 11 July 2021. Retrieved10 July 2021.
- ^"Bekyree- desogestrel and ethinyl estradiol and ethinyl estradiol kit".DailyMed.Archived from the original on 11 July 2021. Retrieved10 July 2021.
- ^"Bimizza 150 microgram/20 microgram Tablets - Summary of Product Characteristics (SmPC)".(emc).Archived from the original on 11 July 2021. Retrieved10 July 2021.
- ^"Caziant Triphasic Regimen- desogestrel and ethinyl estradiol kit".DailyMed.Archived from the original on 11 July 2021. Retrieved10 July 2021.
- ^"Cesia- desogestrel and ethinyl estradiol kit".DailyMed.Archived from the original on 11 July 2021. Retrieved10 July 2021.
- ^"Cimizt 150 microgram/30 microgram Tablets - Summary of Product Characteristics (SmPC)".(emc).Archived from the original on 11 July 2021. Retrieved10 July 2021.
- ^"Cyclessa Tablets (desogestrel and ethinyl estradiol tablets USP)".DailyMed.Archived from the original on 11 July 2021. Retrieved10 July 2021.
- ^"Cyred EQ- desogestrel and ethinyl estradiol kit".DailyMed.Archived from the original on 11 July 2021. Retrieved10 July 2021.
- ^"Desogen Tablets".DailyMed.Archived from the original on 11 July 2021. Retrieved10 July 2021.
- ^"Emoquette- desogestrel and ethinyl estradiol kit".DailyMed.Archived from the original on 11 July 2021. Retrieved10 July 2021.
- ^"Enskyce- desogestrel and ethinyl estradiol kit".DailyMed.Archived from the original on 11 July 2021. Retrieved10 July 2021.
- ^"Isibloom- desogestrel and ethinyl estradiol kit".DailyMed.Archived from the original on 11 July 2021. Retrieved10 July 2021.
- ^"Juleber- desogestrel and ethinyl estradiol kit".DailyMed.Archived from the original on 11 July 2021. Retrieved10 July 2021.
- ^"Kariva- desogestrel/ethinyl estradiol and ethinyl estradiol kit".DailyMed.Archived from the original on 10 July 2021. Retrieved10 July 2021.
- ^"Kimidess (Desogestrel and Ethinyl Estradiol Tablets, USP and Ethinyl Estradiol Tablets, USP), 0.15 mg/0.02 mg and 0.01 mg".DailyMed.Archived from the original on 11 July 2021. Retrieved10 July 2021.
- ^"Marvelon Tablets - Summary of Product Characteristics (SmPC)".(emc).Archived from the original on 10 July 2021. Retrieved10 July 2021.
- ^"Marvelon desogestrel / ethinylestradiol 28 tablets".Therapeutic Goods Administration (TGA).Archived from the original on 2021-07-11. Retrieved2021-07-11.
- ^"Marvelon Product Information".Therapeutic Goods Administration (TGA).Archived from the original on 11 July 2021. Retrieved10 July 2021.
- ^"Mercilon- desogestrel, ethinyl estradiol tablet".DailyMed.Archived from the original on 11 July 2021. Retrieved10 July 2021.
- ^"Mercilon Tablets - Summary of Product Characteristics (SmPC)".(emc).Archived from the original on 10 July 2021. Retrieved10 July 2021.
- ^"Mircette- desogestrel/ethinyl estradiol and ethinyl estradiol kit".DailyMed.Archived from the original on 10 July 2021. Retrieved10 July 2021.
- ^"Ortho-Cept Tablets (Desogestrel And Ethinyl Estradiol)".DailyMed.Archived from the original on 11 July 2021. Retrieved10 July 2021.
- ^"Pimtrea- desogestrel/ethinyl estradiol and ethinyl estradiol kit".DailyMed.Archived from the original on 11 July 2021. Retrieved10 July 2021.
- ^"Reclipsen 28 Day- desogestrel and ethinyl estradiol kit".DailyMed.Archived from the original on 11 July 2021. Retrieved10 July 2021.
- ^"Simliya- desogestrel and ethinyl estradiol and ethinyl estradiol kit".DailyMed.Archived from the original on 11 July 2021. Retrieved10 July 2021.
- ^"Velivet Triphasic Regimen- desogestrel and ethinyl estradiol kit".DailyMed.Archived from the original on 10 July 2021. Retrieved10 July 2021.
- ^"Viorele- desogestrel and ethinyl estradiol and ethinyl estradiol kit".DailyMed.Archived from the original on 11 July 2021. Retrieved10 July 2021.
- ^"Volnea- desogestrel and ethinyl estradiol kit".DailyMed.Archived from the original on 11 July 2021. Retrieved10 July 2021.
- ^Josef Kimmig (14 March 2013).Therapie der Haut- und Geschlechtskrankheiten. Springer-Verlag. pp. 508–.ISBN 978-3-642-94850-3.Archived from the original on 29 August 2021. Retrieved3 June 2019.
- ^"Spezialitäten".Klinische Wochenschrift.30 (15–16): 367. 1952.doi:10.1007/BF01472052.ISSN 0023-2173.S2CID 264011779.
- ^Archived copyArchived 2019-06-09 at theWayback Machine
- ^abHormone und Psyche die Endokrinologie des Alternden Menschen: Fünftes Symposion der Deutschen Gesellschaft für Endokrinologie Freiburg (Breisgau), den 7. bis 9. März 1957. Springer-Verlag. 9 March 2013. pp. 55–.ISBN 978-3-642-87014-9.Archived from the original on 7 April 2022. Retrieved9 June 2019.
|
|---|
Androgens
(incl.AASTooltip anabolic–androgenic steroid) | |
|---|
| Antiandrogens | | ARTooltip Androgen receptorantagonists | |
|---|
Steroidogenesis
inhibitors | |
|---|
| Antigonadotropins | - D2 receptorantagonists (prolactin releasers) (e.g.,domperidone,metoclopramide,risperidone,haloperidol,chlorpromazine,sulpiride)
- Estrogens (e.g.,bifluranol,diethylstilbestrol,estradiol,estradiol esters,ethinylestradiol,ethinylestradiol sulfonate,paroxypropione)
- GnRH agonists (e.g.,leuprorelin)
- GnRH antagonists (e.g.,cetrorelix)
- Progestogens (incl.,chlormadinone acetate,cyproterone acetate,hydroxyprogesterone caproate,gestonorone caproate,medroxyprogesterone acetate,megestrol acetate)
|
|---|
| Others | |
|---|
|
|---|
|
|
|---|
| Estrogens | | ERTooltip Estrogen receptor agonists | - Steroidal:Alfatradiol
- Certainandrogens/anabolic steroids (e.g.,testosterone,testosterone esters,methyltestosterone,metandienone,nandrolone esters) (via estrogenic metabolites)
- Certainprogestins (e.g.,norethisterone,noretynodrel,etynodiol diacetate,tibolone)
- Clomestrone
- Cloxestradiol acetate
- Conjugated estriol
- Conjugated estrogens
- Epiestriol
- Epimestrol
- Esterified estrogens
- Estetrol†
- Estradiol
- Estradiol esters (e.g.,estradiol acetate,estradiol benzoate,estradiol cypionate,estradiol enanthate,estradiol undecylate,estradiol valerate,polyestradiol phosphate,estradiol ester mixtures (Climacteron))
- Estramustine phosphate
- Estriol
- Estriol esters (e.g.,estriol succinate,polyestriol phosphate)
- Estrogenic substances
- Estrone
- Estrone esters
- Ethinylestradiol#
- Hydroxyestrone diacetate
- Mestranol
- Methylestradiol
- Moxestrol
- Nilestriol
- Prasterone (dehydroepiandrosterone; DHEA)
- Promestriene
- Quinestradol
- Quinestrol
|
|---|
| Progonadotropins | |
|---|
|
|---|
| Antiestrogens | ERTooltip Estrogen receptor antagonists
(incl.SERMsTooltip selective estrogen receptor modulators/SERDsTooltip selective estrogen receptor downregulators) | |
|---|
| Aromatase inhibitors | |
|---|
| Antigonadotropins | - Androgens/anabolic steroids (e.g.,testosterone,testosterone esters,nandrolone esters,oxandrolone,fluoxymesterone)
- D2 receptorantagonists (prolactin releasers) (e.g.,domperidone,metoclopramide,risperidone,haloperidol,chlorpromazine,sulpiride)
- GnRH agonists (e.g.,leuprorelin,goserelin)
- GnRH antagonists (e.g.,cetrorelix,elagolix)
- Progestogens (e.g.,chlormadinone acetate,cyproterone acetate,gestonorone caproate,hydroxyprogesterone caproate,medroxyprogesterone acetate,megestrol acetate)
|
|---|
| Others | |
|---|
|
|---|
|
