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Memantine/donepezil

From Wikipedia, the free encyclopedia
Medication

Pharmaceutical compound
Memantine/donepezil
Combination of
MemantineNMDA receptor antagonist
DonepezilAcetylcholinesterase inhibitor
Clinical data
Trade namesNamzaric
AHFS/Drugs.comMicromedex Detailed Consumer Information
License data
Routes of
administration
By mouth
ATC code
Legal status
Legal status
Identifiers
KEGG

Memantine/donepezil, sold under the brand nameNamzaric among others, is afixed dose combination medication used for the treatment ofdementia of theAlzheimer's type.[1] It containsmemantine hydrochloride (it acts as anNMDA receptor antagonist, among various other types of targets like5-HT3 receptor,Nicotinic acetylcholine receptor, andSigma-1 receptor) anddonepezil hydrochloride, which is anacetylcholinesterase inhibitor.[1] It is takenby mouth.[1]

Memantine/donepezil was approved for medical use in the United States in 2014.[3]

References

[edit]
  1. ^abcd"Namzaric- memantine hydrochloride and donepezil hydrochloride capsule; Namzaric- memantine hydrochloride and donepezil hydrochloride kit".DailyMed. 22 January 2019.Archived from the original on 20 January 2022. Retrieved22 December 2023.
  2. ^"Periodic safety update report single assessment donepezil / memantine".European Medicines Agency. 7 March 2024. Retrieved2 May 2024.
  3. ^"Namzaric (memantine hydrochloride extended-release/donepezil hydrochloride) Capsules".U.S.Food and Drug Administration (FDA). 13 May 2015. Archived fromthe original on 22 December 2023. Retrieved22 December 2023.

Further reading

[edit]
Psychoanaleptics: Anti-dementia agents (ATC codeN06D and others)
AChE inhibitor medications
Other medications
ExperimentalBACE inhibitors
Enzyme
(modulators)
ChATTooltip Choline acetyltransferase
AChETooltip Acetylcholinesterase
BChETooltip Butyrylcholinesterase
Transporter
(modulators)
CHTTooltip Choline transporter
VAChTTooltip Vesicular acetylcholine transporter
Release
(modulators)
Inhibitors
Enhancers
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