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| Estrogens | | ERTooltip Estrogen receptor agonists | - Steroidal:Alfatradiol
- Certainandrogens/anabolic steroids (e.g.,testosterone,testosterone esters,methyltestosterone,metandienone,nandrolone esters) (via estrogenic metabolites)
- Certainprogestins (e.g.,norethisterone,noretynodrel,etynodiol diacetate,tibolone)
- Clomestrone
- Cloxestradiol acetate
- Conjugated estriol
- Conjugated estrogens
- Epiestriol
- Epimestrol
- Esterified estrogens
- Estetrol†
- Estradiol
- Estradiol esters (e.g.,estradiol acetate,estradiol benzoate,estradiol cypionate,estradiol enanthate,estradiol undecylate,estradiol valerate,polyestradiol phosphate,estradiol ester mixtures (Climacteron))
- Estramustine phosphate
- Estriol
- Estriol esters (e.g.,estriol succinate,polyestriol phosphate)
- Estrogenic substances
- Estrone
- Estrone esters
- Ethinylestradiol#
- Hydroxyestrone diacetate
- Mestranol
- Methylestradiol
- Moxestrol
- Nilestriol
- Prasterone (dehydroepiandrosterone; DHEA)
- Promestriene
- Quinestradol
- Quinestrol
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| Progonadotropins | |
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| Antiestrogens | ERTooltip Estrogen receptor antagonists (incl.SERMsTooltip selective estrogen receptor modulators/SERDsTooltip selective estrogen receptor downregulators) | |
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| Aromatase inhibitors | |
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| Antigonadotropins | - Androgens/anabolic steroids (e.g.,testosterone,testosterone esters,nandrolone esters,oxandrolone,fluoxymesterone)
- D2 receptorantagonists (prolactin releasers) (e.g.,domperidone,metoclopramide,risperidone,haloperidol,chlorpromazine,sulpiride)
- GnRH agonists (e.g.,leuprorelin,goserelin)
- GnRH antagonists (e.g.,cetrorelix,elagolix)
- Progestogens (e.g.,chlormadinone acetate,cyproterone acetate,gestonorone caproate,hydroxyprogesterone caproate,medroxyprogesterone acetate,megestrol acetate)
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| Others | |
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Androgens (incl.AASTooltip anabolic–androgenic steroid) | |
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| Antiandrogens | | ARTooltip Androgen receptorantagonists | |
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Steroidogenesis inhibitors | |
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| Antigonadotropins | - D2 receptorantagonists (prolactin releasers) (e.g.,domperidone,metoclopramide,risperidone,haloperidol,chlorpromazine,sulpiride)
- Estrogens (e.g.,bifluranol,diethylstilbestrol,estradiol,estradiol esters,ethinylestradiol,ethinylestradiol sulfonate,paroxypropione)
- GnRH agonists (e.g.,leuprorelin)
- GnRH antagonists (e.g.,cetrorelix)
- Progestogens (incl.,chlormadinone acetate,cyproterone acetate,hydroxyprogesterone caproate,gestonorone caproate,medroxyprogesterone acetate,megestrol acetate)
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| Others | |
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