Movatterモバイル変換


[0]ホーム

URL:


Jump to content
WikipediaThe Free Encyclopedia
Search

Acefylline

From Wikipedia, the free encyclopedia
Chemical compound
Pharmaceutical compound
Acefylline
Skeletal formula of acefylline
Ball-and-stick model of the acefylline molecule
Clinical data
Routes of
administration
Intramuscular,Intravenous
ATC code
Identifiers
  • (1,3-Dimethyl-2,6-dioxo-1,2,3,6-tetrahydro-7H-purin-7-yl)acetic acid
CAS Number
PubChemCID
ChemSpider
UNII
ChEMBL
CompTox Dashboard(EPA)
ECHA InfoCard100.010.447Edit this at Wikidata
Chemical and physical data
FormulaC9H10N4O4
Molar mass238.203 g·mol−1
3D model (JSmol)
  • O=C2N(c1ncn(c1C(=O)N2C)CC(=O)O)C
  • InChI=1S/C9H10N4O4/c1-11-7-6(8(16)12(2)9(11)17)13(4-10-7)3-5(14)15/h4H,3H2,1-2H3,(H,14,15) checkY
  • Key:HCYFGRCYSCXKNQ-UHFFFAOYSA-N checkY
  (verify)

Acefylline (INN),[1] also known as7-theophyllineacetic acid, is astimulantdrug of thexanthinechemical class. It acts as anadenosine receptorantagonist. It is combined withdiphenhydramine in thepharmaceuticalpreparationetanautine to help offset diphenhydramine induced drowsiness.[2]

Asilanolmannuronic acid conjugate of acefylline,acefylline methylsilanol mannuronate (INCI; trade nameXantalgosil C) is marketed as alipolyticphosphodiesterase inhibitor. It is used as an ingredient incosmeceuticals for the treatment ofcellulite and as a skin conditioner.[3][4]

See also

[edit]

References

[edit]
  1. ^"International Nonproprietary Names for Pharmaceutical Substances (INN). Recommended International Nonproprietary Names (Rec. INN): List 21"(PDF). World Health Organization. Retrieved29 December 2016.
  2. ^Zuidema J (1978)."Biofarmaceutische en farmacokinetische aspecten van theofylline en acefylline". Thesis (doctoral)--Universiteit van Amsterdam. Archived fromthe original on 2016-12-30. Retrieved2012-09-29.
  3. ^Biosil Technologies (2005)."Xantalgosil C® Datasheet"(PDF). Exsymol S.A.M. Retrieved2022-01-20.
  4. ^Winter, Ruth (2009-10-20).A Consumer's Dictionary of Cosmetic Ingredients (7th ed.). Harmony/Rodale. p. 42.ISBN 9780307459862.
Adrenergics,inhalants
Short-acting β2 agonists
Long-acting β2 agonists
Ultra-long-acting β2 agonists
Other
Glucocorticoids
Anticholinergics/
muscarinic antagonist
Mast cell stabilizers
Xanthines
Eicosanoid inhibition
Leukotriene antagonists
Arachidonate 5-lipoxygenase inhibitors
Thromboxane receptor antagonists
Non-xanthinePDE4 inhibitors
Others/unknown
Combination products
Receptor
(ligands)
P0 (adenine)
P1
(adenosine)
P2
(nucleotide)
P2X
(ATPTooltip Adenosine triphosphate)
P2Y
Transporter
(blockers)
CNTsTooltip Concentrative nucleoside transporters
ENTsTooltip Equilibrative nucleoside transporters
PMATTooltip Plasma membrane monoamine transporter
Enzyme
(inhibitors)
XOTooltip Xanthine oxidase
Others
Others


Stub icon

Thisdrug article relating to therespiratory system is astub. You can help Wikipedia byadding missing information.

Retrieved from "https://en.wikipedia.org/w/index.php?title=Acefylline&oldid=1329174036"
Categories:
Hidden categories:

[8]ページ先頭

©2009-2026 Movatter.jp