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Tranylcypromine/trifluoperazine

From Wikipedia, the free encyclopedia
Combination drug
Pharmaceutical compound
Tranylcypromine/trifluoperaizne
Combination of
TranylcypromineMonoamine oxidase inhibitor
TrifluoperazineTypical antipsychotic
Clinical data
Trade namesParstelin, Parmodalin, Jatrosom N, Stelapar
Routes of
administration
Oral
Legal status
Legal status
  • In general: ℞ (Prescription only)
Identifiers
CAS Number

Tranylcypromine/trifluoperazine (brand namesParstelin,Parmodalin,Jatrosom N,Stelapar) is acombination formulation of themonoamine oxidase inhibitorantidepressant drugtranylcypromine and thetypical antipsychotic drugtrifluoperazine that has been used in the treatment ofmajor depressive disorder.[1][2][3] It contains 10 mg tranylcypromine and 1 mg trifluoperazine.[3][4] The drug has been in clinical use since at least 1961.[3]

It may come to assume a certain place in the treatment ofborderline personality disorder.[5]

See also

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References

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  1. ^Dart RC (2004)."Monoamine Oxidase Inhibitors".Medical Toxicology. Lippincott Williams & Wilkins. pp. 825–.ISBN 978-0-7817-2845-4.
  2. ^Stahl SM (15 May 2014).Prescriber's Guide: Stahl's Essential Psychopharmacology. Cambridge University Press. pp. 783–.ISBN 978-1-107-67502-5.
  3. ^abcStraker M, Grauer H (July 1961)."Clinical Study of a Potent Antidepressant, Tranylcypromine with Trifluorperazine (Parstelin ), in the Aged Chronically Ill".Canadian Medical Association Journal.85 (3):127–130.PMC 1848140.PMID 20326829.
  4. ^Kalinowsky LB, Hippius H, Klein HE (1982).Biological Treatments in Psychiatry. Grune and Stratton, Harcourt Brace Jovanovich.ISBN 978-0-8089-1423-5.
  5. ^Cowdry, R. W., & Gardner, D. L. (1988). Pharmacotherapy of borderline personality disorder. Alprazolam, carbamazepine, trifluoperazine, and tranylcypromine. Archives of general psychiatry, 45(2), 111–119.https://doi.org/10.1001/archpsyc.1988.01800260015002
SSRIsTooltip Selective serotonin reuptake inhibitors
SNRIsTooltip Serotonin–norepinephrine reuptake inhibitors
NRIsTooltip Norepinephrine reuptake inhibitors
NDRIsTooltip Norepinephrine–dopamine reuptake inhibitors
NaSSAsTooltip Noradrenergic and specific serotonergic antidepressants
SARIsTooltip Serotonin antagonist and reuptake inhibitors
SMSTooltip Serotonin modulator and stimulators
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TCAsTooltip Tricyclic antidepressants
TeCAsTooltip Tetracyclic antidepressants
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Non-selective
MAOATooltip Monoamine oxidase A-selective
MAOBTooltip Monoamine oxidase B-selective
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