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Selective PPAR modulator

From Wikipedia, the free encyclopedia
(Redirected fromSelective PPARγ modulator)

Aselective PPAR modulator (SPPARM) is aselective receptor modulator of theperoxisome proliferator-activated receptor (PPAR).[1][2][3] Examples include SPPARMs of thePPARγ,BADGE,EPI-001,INT-131,MK-0533, andS26948.

See also

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References

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  1. ^Fruchart, Jean-Charles; Santos, Raul D.; Aguilar-Salinas, Carlos; Aikawa, Masanori; Al Rasadi, Khalid; Amarenco, Pierre; Barter, Philip J.; Ceska, Richard; Corsini, Alberto; Després, Jean-Pierre; Duriez, Patrick; Eckel, Robert H.; Ezhov, Marat V.; Farnier, Michel; Ginsberg, Henry N.; Hermans, Michel P.; Ishibashi, Shun; Karpe, Fredrik; Kodama, Tatsuhiko; Koenig, Wolfgang; Krempf, Michel; Lim, Soo; Lorenzatti, Alberto J.; McPherson, Ruth; Nuñez-Cortes, Jesus Millan; Nordestgaard, Børge G.; Ogawa, Hisao; Packard, Chris J.; Plutzky, Jorge; Ponte-Negretti, Carlos I.; Pradhan, Aruna; Ray, Kausik K.; Reiner, Željko; Ridker, Paul M.; Ruscica, Massimiliano; Sadikot, Shaukat; Shimano, Hitoshi; Sritara, Piyamitr; Stock, Jane K.; Su, Ta-Chen; Susekov, Andrey V.; Tartar, André; Taskinen, Marja-Riitta; Tenenbaum, Alexander; Tokgözoğlu, Lale S.; Tomlinson, Brian; Tybjærg-Hansen, Anne; Valensi, Paul; Vrablík, Michal; Wahli, Walter; Watts, Gerald F.; Yamashita, Shizuya; Yokote, Koutaro; Zambon, Alberto; Libby, Peter (4 June 2019)."The selective peroxisome proliferator-activated receptor alpha modulator (SPPARMα) paradigm: conceptual framework and therapeutic potential".Cardiovascular Diabetology.18 (1): 71.doi:10.1186/s12933-019-0864-7.ISSN 1475-2840.PMC 6549355.PMID 31164165.
  2. ^Fruchart, Jean-Charles; Hermans, Michel P.; Fruchart-Najib, Jamila; Kodama, Tatsuhiko (3 January 2021)."Selective Peroxisome Proliferator-Activated Receptor Alpha Modulators (SPPARMα) in the Metabolic Syndrome: Is Pemafibrate Light at the End of the Tunnel?".Current Atherosclerosis Reports.23 (1): 3.doi:10.1007/s11883-020-00897-x.ISSN 1534-6242.PMC 7779417.PMID 33392801.
  3. ^Balint, B. L.; Nagy, L. (March 2006). "Selective modulators of PPAR activity as new therapeutic tools in metabolic diseases".Endocrine, Metabolic & Immune Disorders Drug Targets.6 (1):33–43.doi:10.2174/187153006776056620.ISSN 1871-5303.PMID 16611163.


PPARTooltip Peroxisome proliferator-activated receptormodulators
PPARαTooltip Peroxisome proliferator-activated receptor alpha
PPARδTooltip Peroxisome proliferator-activated receptor delta
PPARγTooltip Peroxisome proliferator-activated receptor gamma
Non-selective


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