Movatterモバイル変換

Jump to content

List of corticosteroid esters

Bahasa Melayu

From Wikipedia, the free encyclopedia

Beclometasone dipropionate, an example of a widely used corticosteroid ester. Note thepropionate groups at the C17α and C21α positions (top right corner).

This is alist ofcorticosteroid esters, includingesters ofsteroidal glucocorticoids andmineralocorticoids.^[1]^[2]^[3]

Esters of natural corticosteroids

Desoxycortone esters

See also:11-Deoxycorticosterone andDesoxycortone

Desoxycortone acetate (deoxycortone acetate; desoxycorticosterone acetate)
Desoxycortone cypionate (deoxycortone cypionate; desoxycorticosterone cypionate)^[4]
Desoxycortone enanthate (deoxycortone enanthate; deoxycorticosterone enanthate)
Desoxycortone glucoside (deoxycortone glucoside; deoxycorticosterone glucoside)
Desoxycortone pivalate (deoxycortone pivalate; deoxycorticosterone pivalate)

Hydrocortisone esters

See also:Cortisol andHydrocortisone

Benzodrocortisone (hydrocortisone 17-benzoate)
Hydrocortamate (hydrocortisone 21-(diethylamino)acetate)
Hydrocortisone aceponate (hydrocortisone 21-acetate 17α-propionate)
Hydrocortisone acetate
Hydrocortisone bendazac
Hydrocortisone buteprate (hydrocortisone 17α-butyrate 21-propionate)
Hydrocortisone butyrate (hydrocortisone 17α-butyrate)
Hydrocortisone 21-butyrate
Hydrocortisone cypionate (hydrocortisone cyclopentanepropionate)
Hydrocortisone phosphate
Hydrocortisone succinate (hydrocortisone hemisuccinate)
Hydrocortisone tebutate
Hydrocortisone valerate
Hydrocortisone xanthogenic acid

Esters of other natural corticosteroids

See also:11-Dehydrocorticosterone,11-Deoxycortisol,Cortodoxone,Cortisone, andCorticosterone

11-Dehydrocorticosterone acetate
Cortifen (cortodoxone chlorphenacyl ester)
Cortisone acetate
Corticosterone acetate
Corticosterone benzoate
Cortodoxone acetate

Esters of synthetic corticosteroids

Beclometasone esters

See also:Beclometasone

Beclometasone dipropionate (beclomethasone dipropionate)
Beclometasone salicylate
Beclometasone valeroacetate

Betamethasone esters

See also:Betamethasone

Betamethasone acetate
Betamethasone acibutate (betamethasone 21-acetate 17α-isobutyrate)
Betamethasone adamantoate
Betamethasone benzoate
Betamethasone dipropionate
Betamethasone divalerate
Betamethasone phosphate (betamethasone phosphate)
Betamethasone succinate
Betamethasone valerate
Betamethasone valeroacetate (betamethasone 21-acetate 17α-valerate)
Cortobenzolone (betamethasone salicylate)

Clocortolone esters

See also:Clocortolone

Dexamethasone esters

See also:Dexamethasone

Fluocinolone acetonide esters

See also:Fluocinolone acetonide

Ciprocinonide (fluocinolone acetonide cyclopropylcarboxylate)
Fluocinonide (fluocinolone acetonide 21-acetate)
Procinonide (fluocinolone acetonide propionate)

Fluocortolone esters

See also:Fluocortolone

Fluocortin (fluocortolone-21-carboxylate)
Fluocortin butyl (fluocortolone-21-carboxylate 21-butylate)
Fluocortolone caproate
Fluocortolone pivalate

Fluprednisolone esters

See also:Fluprednisolone

Fluprednisolone acetate
Fluprednisolone succinate (fluprednisolone hemisuccinate)
Fluprednisolone valerate

Methylprednisolone esters

See also:Methylprednisolone

Methylprednisolone aceponate
Methylprednisolone acetate
Methylprednisolone cyclopentylpropionate
Methylprednisolone phosphate
Methylprednisolone succinate (methylprednisolone hemisuccinate)
Methylprednisolone suleptanate

Prednisolone esters

See also:Prednisolone

Prednazate (prednisolone succinate andperphenazine compound)
Prednazoline (prednisolone phosphate andfenoxazoline compound)
Prednicarbate (prednisolone 17-(ethyl carbonate) 21-propionate)
Prednimustine (prednisolonechlorambucil ester)
Prednisolamate (prednisolone diethylaminoacetate)
Prednisolone acetate
Prednisolone hexanoate
Prednisolone metasulphobenzoate (prednisolone 21-(3-sulfobenzoate))
Prednisolone palmitate
Prednisolone phosphate
Prednisolone piperidinoacetate
Prednisolone pivalate
Prednisolone steaglate (prednisolone stearoyl-glycolate)
Prednisolone stearoylglycolate
Prednisolone succinate (prednisolone hemisuccinate)
Prednisolone sulfate
Prednisolone tebutate (prednisolonetert-butylacetate)
Prednisolone tetrahydrophthalate
Prednisolone valerate
Prednisolone valeroacetate

Prednisone esters

See also:Prednisone

Tixocortol esters

See also:Tixocortol

Butixocort (tixocortol butyrate)
Butixocort propionate (tixocortol butyrate propionate)
Tixocortol pivalate

Triamcinolone acetonide esters

See also:Triamcinolone acetonide

Flupamesone (triamcinolone acetonide metembonate)
Triamcinolone acetonide phosphate
Triamcinolone acetonide succinate (triamcinolone acetonide hemisuccinate)
Triamcinolone benetonide (triamcinolone acetonide 21-(benzoyl-β-aminoisobutyrate))
Triamcinolone furetonide (triamcinolone acetonide 21-(2-benzofurancarboxylate))
Triamcinolone hexacetonide (triamcinolone acetonide 21-(tert-butylacetate))

Esters of other synthetic corticosteroids

Δ⁷-Prednisolone 21-acetate
Alclometasone dipropionate
Amcinonide (triamcinolone acetate cyclopentanonide)
Chloroprednisone acetate
Ciclometasone (a corticosteroid 21-[4-[(acetylamino)methyl]cyclohexyl]carboxylate ester)
Clobetasol propionate
Clobetasone butyrate
Cloprednol acetate
Cormetasone acetate
Cortivazol (a corticosteroid 21-acetate ester)
Cloticasone propionate
Deflazacort (a corticosteroid 21-acetate ester)
Deprodone propionate
Desonide phosphate
Desonide pivalate
Dichlorisone acetate
Dichlorisone diacetate
Diflorasone diacetate
Diflucortolone pivalate
Diflucortolone valerate
Difluprednate (difluoroprednisolone butyrate acetate)
Dimesone acetate
Drocinonide phosphate
Etiprednol dicloacetate
Fluazacort (a corticosteroid 21-acetate ester)
Fludrocortisone acetate
Flumetasone acetate
Flumetasone pivalate
Flunisolide acetate
Fluorometholone acetate
Fluperolone acetate
Fluprednidene acetate
Fluticasone furoate
Fluticasone propionate
Formocortal (a corticosteroid 21-acetate ester)
Halopredone acetate (halopredone diacetate)
Icometasone enbutate
Isoflupredone acetate
Locicortolone dicibate
Loteprednol etabonate
Meclorisone dibutyrate
Meprednisone acetate
Meprednisone succinate (meprednisone hemisuccinate)
Mometasone furoate
Nicocortonide (a corticosteroid 21-isonicotinate ester)
Nicocortonide acetate
Paramethasone acetate
Paramethasone phosphate
Prebediolone acetate
Prednylidene diethylaminoacetate
Rofleponide palmitate
Ticabesone propionate
Timobesone acetate
Triamcinolone aminobenzal benzamidoisobutyrate
Triamcinolone diacetate
Ulobetasol propionate (halobetasol propionate)

See also

References

^J. Elks (14 November 2014).The Dictionary of Drugs: Chemical Data: Chemical Data, Structures and Bibliographies. Springer.ISBN 978-1-4757-2085-3.
^Index Nominum 2000: International Drug Directory. Taylor & Francis. 2000.ISBN 978-3-88763-075-1.
^"The use of stems in the selection of International Nonproprietary Names (INN) for pharmaceutical substances"(PDF). WHO. 2013.
^J. Elks (14 November 2014).The Dictionary of Drugs: Chemical Data: Chemical Data, Structures and Bibliographies. Springer. pp. 665–.ISBN 978-1-4757-2085-3.

v
t
e

Glucocorticoids andantiglucocorticoids (D07,H02)

Glucocorticoids

Cortisol-like and related (16-unsubstituted):Chloroprednisone
Cloprednol
Difluprednate
Fludrocortisone
Flugestone acetate (flurogestone acetate)
Fluocinolone
Fluorometholone
- Fluorometholone acetate
Fluperolone
- Fluperolone acetate
Fluprednisolone
- Fluprednisolone esters
Loteprednol (+tobramycin)
Medrysone
Methylprednisolone
- Methylprednisolone esters
Methylprednisolone aceponate
Prednicarbate
Prednisolone^#
Prednisone
Tixocortol
- Tixocortol pivalate

Methasones and related (16-substituted):Alclometasone
Beclometasone
- Beclometasone esters
Betamethasone^#
- Betamethasone esters
Clobetasol
- Clobetasol propionate
Clobetasone
Clocortolone
- Clocortolone esters
Cortivazol
Desoximetasone
Dexamethasone^#
- Dexamethasone esters
Diflorasone
Diflucortolone
- Diflucortolone valerate
Fluclorolone
Flumetasone
Fluocortin
Fluocortolone
- Fluocortolone esters
Fluprednidene acetate
Fluticasone
- Fluticasone furoate
- Fluticasone propionate
Halometasone
Meprednisone
Mometasone
- Mometasone furoate
Paramethasone
Prednylidene
Rimexolone
Triamcinolone
Ulobetasol (halobetasol)

Antiglucocorticoids

Synthesis modifiers

^#WHO-EM
^‡Withdrawn from market
Clinical trials:
- ^†Phase III
- ^§Never to phase III

See also: Glucocorticoid receptor modulators; Mineralocorticoids and antimineralocorticoids; List of corticosteroids

v t e Mineralocorticoids andantimineralocorticoids (H02)
Mineralocorticoids	Desoxycortone (desoxycorticosterone) Desoxycortone esters Hydrocortisone (cortisol) Hydrocortisone esters Fludrocortisone Fludrocortisone acetate Methylprednisolone Methylprednisolone esters Prednisolone Prednisolone esters Prednisone Prednisone esters
Antimineralocorticoids	Steroidal:Canrenoate potassium (potassium canrenoate) Canrenone Drospirenone Dydrogesterone Eplerenone Gestodene Medrogestone Progesterone Spironolactone Trimegestone Nonsteroidal:Amlodipine Apararenone^§ Benidipine Esaxerenone^† Felodipine Finerenone Nifedipine Nimodipine Nitrendipine
Synthesis modifiers	Acetoxolone Aminoglutethimide Carbenoxolone Enoxolone Ketoconazole Metyrapone Mitotane Trilostane
^#WHO-EM ^‡Withdrawn from market Clinical trials: ^†Phase III ^§Never to phase III See also Mineralocorticoid receptor modulators Glucocorticoids and antiglucocorticoids List of corticosteroids

v
t
e

Glucocorticoid receptor modulators

GRTooltip Glucocorticoid receptor

Agonists	Cortisol-like and related (16-unsubstituted):3α,5α-Tetrahydrocorticosterone 5α-Dihydrocorticosterone 9α-Fluorocortisone (alfluorone) 11-Dehydrocorticosterone (11-oxocorticosterone, 17-deoxycortisone) 11-Dehydrocorticosterone acetate 11-Deoxycorticosterone (desoxycortone, deoxycortone, desoxycorticosterone) Desoxycortone esters 11-Deoxycortisol (cortodoxone, cortexolone) Cortifen (cortiphen, kortifen) Cortodoxone acetate 21-Deoxycortisol Δ⁷-Prednisolone Δ⁷-Prednisolone 21-acetate Amebucort Chloroprednisone Chloroprednisone acetate Cloprednol Cloprednol acetate Corticosterone Corticosterone acetate Corticosterone benzoate Cortisol (hydrocortisone) Benzodrocortisone (hydrocortisone benzoate) Hydrocortamate (hydrocortisone diethylaminoacetate) Hydrocortisone esters Cortisone Cortisone acetate Deprodone Deprodone propionate Dichlorisone Dichlorisone acetate Dichlorisone diacetate Difluprednate Endrisone (endrysone) Etiprednol Etiprednol dicloacetate (etiprednol dichloroacetate) Fludrocortisone (fludrocortone) Fludrocortisone acetate Fluorometholone Fluorometholone acetate Fluperolone Fluperolone acetate Fluprednisolone Fluprednisolone esters Halopredone Halopredone acetate (halopredone diacetate) Isoflupredone (9α-fluoroprednisolone) Isoflupredone acetate Loteprednol Mazipredone (depersolone) Medrysone Methylprednisolone Methylprednisolone esters Prebediolone Prebediolone acetate Prednisolone Prednazate Prednazoline Prednicarbate (prednisolone ethylcarbonate propionate) Prednimustine Prednisolamate (prednisolone diethylaminoacetate) Prednisolone esters Prednisone Prednisone esters Pregnenolone Pregnenolone acetate Pregnenolone succinate (pregnenolone hemisuccinate) Resocortol Tipredane Tixocortol Butixocort (tixocortol butyrate) Butixocort propionate Tixocortol pivalate Methasones and related (16-substituted):16α-Methyl-11-oxoprednisolone Alclometasone Alclometasone dipropionate Amelometasone Beclometasone (beclomethasone) Beclometasone esters Betamethasone (betametasone) Betamethasone esters Cortobenzolone (betamethasone salicylate) Ciclometasone (ciclomethasone, cyclomethasone) Clobetasol Clobetasol propionate Clobetasone Clobetasone butyrate Clocortolone Clocortolone esters Cloticasone Cloticasone propionate Cormetasone (cormethasone) Cormetasone acetate Descinolone Desoximetasone (desoxymethasone) Dexamethasone (dexametasone) Dexamethasone esters Diflorasone Diflorasone diacetate Diflucortolone Diflucortolone pivalate Diflucortolone valerate Dimesone Dimesone acetate Doxibetasol (doxybetasol) Fluclorolone Flumetasone (flumethasone) Flumetasone acetate Flumetasone pivalate Fluocinolone Fluocortin Fluocortin butyl (fluocortin butylate) Fluocortolone Fluocortolone esters Fluprednidene (fluprednylidene) Fluprednidene acetate Fluticasone Fluticasone furoate Fluticasone propionate Halocortolone Halometasone Icometasone Icometasone enbutate (icometasone butyrate acetate) Isoprednidene Locicortolone (locicortone) Locicortolone dicibate (locicortone dicibate) Meclorisone Meclorisone dibutyrate Meprednisone (methylprednisone) Meprednisone acetate Meprednisone hydrogen succinate (methylprednisone hemisuccinate) Mometasone Mometasone furoate Paramethasone Paramethasone acetate Paramethasone disodium phosphate Paramethasone phosphate Prednylidene Prednylidene diethylaminoacetate Rimexolone Ticabesone Ticabesone propionate Timobesone Timobesone acetate Triamcinolone Triamcinolone diacetate Ulobetasol (halobetasol) Ulobetasol propionate Vamorolone Cyclic ketals (16,17-cyclized):Acrocinonide (triamcinolone acroleinide) Amcinafal (triamcinolone pentanonide) Amcinafide (triamcinolone acetophenide) Amcinonide (triamcinolone acetate cyclopentanonide) Budesonide Ciclesonide Cicortonide Deflazacort (azacort) Descinolone acetonide Desonide (hydroxyprednisolone acetonide) Desonide disodium phosphate Desonide pivalate Dexbudesonide Drocinonide Drocinonide phosphate Fluazacort Fluclorolone acetonide (flucloronide) Fludroxycortide (flurandrenolone, flurandrenolide) Flumoxonide Flunisolide Flunisolide acetate Fluocinolone acetonide Ciprocinonide (fluocinolone acetonide cyclopropylcarboxylate) Fluocinonide (fluocinolide, fluocinolone acetonide acetate) Procinonide (fluocinolone acetonide propionate) Formocortal Halcinonide Itrocinonide Rofleponide Rofleponide palmitate Tralonide Triamcinolone acetonide Flupamesone (triamcinolone acetonide metembonate) Triamcinolone acetonide esters Triamcinolone aminobenzal benzamidoisobutyrate (TBI-PAB) Triclonide Others/atypical (other expanded steroid ring systems, homosteroids, and non-pregnane steroids):Cortisuzol Cortivazol Domoprednate Naflocort Nicocortonide Nicocortonide acetate Nivacortol (nivazol) Oxisopred RU-26988 RU-28362 Non-corticosteroids with some glucocorticoid activity:15β-Hydroxycyproterone acetate 17α-Hydroxyprogesterone Bromoketoprogesterone Chlormadinone acetate Cyproterone Cyproterone acetate Danazol Delmadinone acetate Desogestrel DU-41165 Etonogestrel Flugestone Flugestone acetate (flurogestone acetate) Fluoromedroxyprogesterone acetate Fluoxymesterone Gestodene Medrogestone Medroxyprogesterone acetate Megestrol acetate Metribolone Norgestomet Osaterone acetate Progesterone Promegestone RU-2309 Quingestrone Segesterone acetate (nestorone) Tetrahydrogestrinone Nonsteroidal glucocorticoids:AZD-5423 GSK-9027
Mixed (SEGRMsTooltip Selective glucocorticoid receptor agonists)	Dagrocorat Fosdagrocorat Mapracorat
Antagonists	7α-Hydroxy-DHEA 17α-Methylprogesterone Aglepristone Asoprisnil Asoprisnil ecamate C108297 C113176 CORT-108297 Cyproterone acetate Dazucorilant Exicorilant (CORT-125281) Guggulsterone Ketoconazole Lilopristone LLY-2707 Metapristone (RU-42633) Miconazole Mifepristone (RU-486) Miricorilant (CORT-118335) Onapristone ORG-34116 ORG-34517 (SCH-900636) ORG-34850 Pregnenolone 16α-carbonitrile Relacorilant (CORT-125134) RTI 3021–012 RTI 3021–022 Telapristone Tibolone Toripristone Ulipristal acetate Zavacorilant
Others	Antisense oligonucleotides:IONIS-GCCR_Rx (ISIS-426115)

See also: Receptor/signaling modulators; Glucocorticoids and antiglucocorticoids; Mineralocorticoid receptor modulators; List of corticosteroids

v
t
e

Mineralocorticoid receptor modulators

MRTooltip Mineralocorticoid receptor

Agonists

Antagonists

See also: Receptor/signaling modulators; Mineralocorticoids and antimineralocorticoids; Glucocorticoid receptor modulators; List of corticosteroids

Retrieved from "https://en.wikipedia.org/w/index.php?title=List_of_corticosteroid_esters&oldid=1188034274"

Hidden categories:

[8]ページ先頭

©2009-2025 Movatter.jp