| Ionotropic | | GABAATooltip γ-Aminobutyric acid A receptor | - Positive modulators (abridged; seehere for a full list):α-EMTBL
- Alcohols (e.g.,drinking alcohol,2M2B)
- Anabolic steroids
- Avermectins (e.g.,ivermectin)
- Barbiturates (e.g.,phenobarbital)
- Benzodiazepines (e.g.,diazepam)
- Bromide compounds (e.g.,potassium bromide)
- Carbamates (e.g.,meprobamate)
- Carbamazepine
- Chloralose
- Chlormezanone
- Clomethiazole
- Dihydroergolines (e.g.,ergoloid (dihydroergotoxine))
- Etazepine
- Etifoxine
- Fenamates (e.g.,mefenamic acid)
- Flavonoids (e.g.,apigenin,hispidulin)
- Fluoxetine
- Flupirtine
- Imidazoles (e.g.,etomidate)
- Kava constituents (e.g.,kavain)
- Lanthanum
- Loreclezole
- Monastrol
- Neuroactive steroids (e.g.,allopregnanolone,cholesterol,THDOC)
- Niacin
- Niacinamide
- Nonbenzodiazepines (e.g.,β-carbolines (e.g.,abecarnil),cyclopyrrolones (e.g.,zopiclone),imidazopyridines (e.g.,zolpidem),pyrazolopyrimidines (e.g.,zaleplon))
- Norfluoxetine
- Petrichloral
- Phenols (e.g.,propofol)
- Phenytoin
- Piperidinediones (e.g.,glutethimide)
- Propanidid
- Pyrazolopyridines (e.g.,etazolate)
- Quinazolinones (e.g.,methaqualone)
- Retigabine (ezogabine)
- ROD-188
- Skullcap constituents (e.g.,baicalin)
- Stiripentol
- Sulfonylalkanes (e.g.,sulfonmethane (sulfonal))
- Topiramate
- Valerian constituents (e.g.,valerenic acid)
- Volatiles/gases (e.g.,chloral hydrate,chloroform,diethyl ether,paraldehyde,sevoflurane)
- Negative modulators:1,3M1B
- 3M2B
- 11-Ketoprogesterone
- 17-Phenylandrostenol
- α3IA
- α5IA (LS-193,268)
- β-CCB
- β-CCE
- β-CCM
- β-CCP
- β-EMGBL
- Anabolic steroids
- Amiloride
- Anisatin
- β-Lactams (e.g.,penicillins,cephalosporins,carbapenems)
- Basmisanil
- Bemegride
- Bicyclic phosphates (TBPS,TBPO,IPTBO)
- BIDN
- Bilobalide
- Bupropion
- CHEB
- Chlorophenylsilatrane
- Cicutoxin
- Cloflubicyne
- Cyclothiazide
- DHEA
- DHEA-S
- Dieldrin
- (+)-DMBB
- DMCM
- DMPC
- EBOB
- Etbicyphat
- FG-7142 (ZK-31906)
- Fiproles (e.g.,fipronil)
- Flavonoids (e.g.,amentoflavone,oroxylin A)
- Flumazenil
- Fluoroquinolones (e.g.,ciprofloxacin)
- Flurothyl
- Furosemide
- Golexanolone
- Iomazenil (123I)
- IPTBO
- Isopregnanolone (sepranolone)
- L-655,708
- Laudanosine
- Lindane
- MaxiPost
- Morphine
- Morphine-3-glucuronide
- MRK-016
- Naloxone
- Naltrexone
- Nicardipine
- Nonsteroidal antiandrogens (e.g.,apalutamide,bicalutamide,enzalutamide,flutamide,nilutamide)
- Oenanthotoxin
- Pentylenetetrazol (pentetrazol)
- Phenylsilatrane
- Picrotoxin (i.e.,picrotin,picrotoxinin anddihydropicrotoxinin)
- Pregnenolone sulfate
- Propybicyphat
- PWZ-029
- Radequinil
- Ro 15-4513
- Ro 19-4603
- RO4882224
- RO4938581
- Sarmazenil
- SCS
- Suritozole
- TB-21007
- TBOB
- TBPS
- TCS-1105
- Terbequinil
- TETS
- Thujone
- U-93631
- Zinc
- ZK-93426
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| GABAA-ρTooltip γ-Aminobutyric acid A-rho receptor | |
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