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Cannabinoidergic

From Wikipedia, the free encyclopedia
Working on the endocannabinoid neurotransmitters

Cannabinoidergic, orcannabinergic, means "working on theendocannabinoidneurotransmitters". As with terms such asdopaminergic andserotonergic, related proteins and cellular components involved in endocannabinoid signaling, such as thecannabinoid (CB1) receptor, as well as exogenous compounds, such asphytocannabinoids or othercannabinoids which modulate the activity ofendocannabinoid system, can be described ascannabinoidergic.[1]

See also

[edit]

References

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  1. ^Palmer, SL; Thakur GA;Makriyannis A (December 31, 2002). "Cannabinergic ligands".Chemistry and Physics of Lipids.121 (1–2):3–19.doi:10.1016/s0009-3084(02)00143-3.PMID 12505686.


Receptor
(ligands)
CB1Tooltip Cannabinoid receptor type 1
Agonists
(abridged,
full list)
Inverse agonists
Antagonists
CB2Tooltip Cannabinoid receptor type 2
Agonists
Antagonists
NAGly
(
GPR18)
Agonists
Antagonists
GPR55
Agonists
Antagonists
GPR119
Agonists
Transporter
(modulators)
eCBTsTooltip Endocannabinoid transporter
Enzyme
(modulators)
FAAHTooltip Fatty acid amide hydrolase
MAGL
ABHD6
ABHD12
Others
  • Others:2-PG(directly potentiates activity of 2-AG at CB1 receptor)
  • ARN-272(FAAH-like anandamide transporter inhibitor)
See also
Receptor/signaling modulators
Cannabinoids (cannabinoids by structure)


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