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| Formula | C17H24Cl2N2 |
| Molar mass | 327.29 g·mol−1 |
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BD1052 orN-[2-(3,4-dichlorophenyl)ethyl]-N-2-propen-1-yl-1-pyrrolidineethanamine is a selectivesigma receptoragonist, with a reportedbinding affinity ofKi = 2 ± 0.5 nM for thesigma-1 receptor and 30 times selectivity over thesigma-2 receptor.[1]
Consistent with other reportedsigma receptoragonists, pretreating Swiss Webster mice with BD1052 significantly increases the behavioral toxicity of cocaine.[1]
